SCHEMBL9842959

SCHEMBL9842959

O=C(Nc1ccccc1O)c1cnoc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.54
RAB9A P51151 3/20 0.54
MEN1 O00255 3/20 0.54
KMT2A Q03164 3/20 0.54
TP53 P04637 2/20 0.54
GAA P10253 2/20 0.51
LMNA P02545 1/20 0.51
HTT P42858 1/20 0.51
RPS6KA3 P51812 1/20 0.49
TOP1 P11387 2/20 0.46
TOP2A P11388 1/20 0.46
TOP2B Q02880 1/20 0.46
METAP2 P50579 1/20 0.45
TERT O14746 1/20 0.45
HDAC1 Q13547 1/20 0.45
MAOB P27338 1/20 0.45
POLB P06746 1/20 0.45
ALDH1A1 P00352 1/20 0.44
AURKA O14965 1/20 0.41
KCNMA1 Q12791 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL892704 0.79 HTT (0.54) NPC1RAB9AMEN1KMT2AHTT
SCHEMBL6029925 0.77 NPC1 (0.82) NPC1RAB9AMEN1KMT2ATP53
SCHEMBL4946074 0.76 NPC1 (0.73) NPC1RAB9AMEN1KMT2ATP53
SCHEMBL1470784 0.76 NPC1 (0.73) NPC1RAB9AMEN1KMT2ATP53
SCHEMBL9842945 0.74 HSD17B2 (0.38) NPC1RAB9AMEN1KMT2ATP53
SCHEMBL9842954 0.74 NQO2 (0.54) NPC1RAB9AMEN1KMT2ATP53
SCHEMBL18086516 0.73 RAB9A (0.68) NPC1RAB9AMEN1KMT2ATP53
SCHEMBL9081513 0.73 TRPV1 (0.50) NPC1RAB9AMEN1KMT2AGAA
SCHEMBL1520536 0.73 HDAC1 (0.70) TP53GAALMNAHTTHDAC1
SCHEMBL462324 0.73 MEN1 (0.66) NPC1RAB9AMEN1KMT2ATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0440503-A1 4-Isoxazolecarboxamide derivatives SYNTEX (U.S.A.) INC. (US) 1991-08-07 EP disclosed