SCHEMBL9843434

SCHEMBL9843434

O=c1nc2ccc(Cc3ccccc3)nc2nc2ncccc12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 8/20 0.41
PDE4A P27815 1/20 0.41
PDE4B Q07343 1/20 0.41
PDE4C Q08493 1/20 0.41
PDE4D Q08499 1/20 0.41
KMT2A Q03164 2/20 0.40
MEN1 O00255 1/20 0.40
ELANE P08246 1/20 0.40
F2 P00734 1/20 0.38
F10 P00742 1/20 0.38
F7 P08709 1/20 0.38
F3 P13726 1/20 0.38
FEN1 P39748 1/20 0.36
MET P08581 1/20 0.36
IDO1 P14902 1/20 0.36
TSHR P16473 1/20 0.36
HIF1A Q16665 1/20 0.36
PAX8 Q06710 1/20 0.35
ALDH1A1 P00352 1/20 0.35
NPC1 O15118 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2693525 0.76 HCAR2 (0.42) HCAR2F2F10F7F3
SCHEMBL9843440 0.75 PAX8 (0.45) HCAR2PDE4APDE4BPDE4CPDE4D
SCHEMBL30276684 0.75 IDO1 (0.38) HCAR2PDE4APDE4BPDE4CPDE4D
SCHEMBL8967704 0.73 CYP3A4 (0.46) HCAR2F2F10F7F3
SCHEMBL1650848 0.72 PLAUR (0.47) HCAR2KMT2AMEN1F2F10
Hydrochloric Acid SCHEMBL5336924 0.70 PLAUR (0.46) HCAR2KMT2AMEN1F2F10
SCHEMBL22762116 0.70 ALDH1A1 (0.45) KMT2AMEN1ELANEALDH1A1
SCHEMBL8749880 0.69 BRD4 (0.45) FEN1METPAX8ALDH1A1
Quinoline SCHEMBL28178121 0.65 ALDH1A1 (0.57) ALDH1A1NPC1RAB9A
SCHEMBL15301760 0.63 CCR1 (0.55) TSHRHIF1APAX8ALDH1A1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0429987-A2 5,11-Dihydro-6H-dipyrido[3,2-b:2',3'-e] [1,4]diazepines and their use in the prevention or treatment of HIV infection BOEHRINGER INGELHEIM PHARMACEUTICALS INC. (US) 1991-06-05 EP disclosed