SCHEMBL9844802

SCHEMBL9844802

Nc1nc(O)c2c(CCc3ccc(C(=O)O)cc3)c(Br)n(Cc3ccccc3)c2n1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 3/20 0.40
AGTR2 P50052 3/20 0.40
TLR7 Q9NYK1 2/20 0.38
PPARG P37231 1/20 0.38
FOLH1 Q04609 1/20 0.38
KDM4E B2RXH2 1/20 0.37
MEN1 O00255 1/20 0.37
USP2 O75604 1/20 0.37
ALDH1A1 P00352 1/20 0.37
POLB P06746 1/20 0.37
GAA P10253 1/20 0.37
MAPT P10636 1/20 0.37
THRB P10828 1/20 0.37
NR4A1 P22736 1/20 0.37
APEX1 P27695 1/20 0.37
APOBEC3A P31941 1/20 0.37
RECQL P46063 1/20 0.37
KMT2A Q03164 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
HIF1A Q16665 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9844856 0.80 DHFR (0.43) KDM4EALDH1A1L3MBTL1
SCHEMBL9844852 0.80 DHFR (0.43) KDM4EALDH1A1L3MBTL1
Butane SCHEMBL9844926 0.79 DHFR (0.40)
SCHEMBL9844931 0.78 ALDH1A1 (0.39) KDM4EMEN1ALDH1A1GAAMAPT
SCHEMBL9844747 0.73 CCR6 (0.45) TLR7ALDH1A1SMN1; SMN2HIF1ADRD2
SCHEMBL9844768 0.70 TBXAS1 (0.39) MEN1ALDH1A1MAPTKMT2AMBOAT4
SCHEMBL27709073 0.67 MBOAT4 (0.50) ALDH1A1POLBMAPTKMT2ATDP1
SCHEMBL9046718 0.66 TYMS (0.54) MBOAT4
SCHEMBL8801558 0.66 MBOAT4 (0.44) KDM4EALDH1A1POLBMAPTKMT2A
SCHEMBL1926270 0.66 HDAC1 (0.64) ALDH1A1NR4A1HDAC1HDAC8PPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0438261-A2 Condensed heterocyclic glutamic acid derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1991-07-24 EP claimed
EP-0438261-A2 Condensed heterocyclic glutamic acid derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1991-07-24 EP disclosed