SCHEMBL9844778

SCHEMBL9844778

Nc1nc(O)c2c(CCc3ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)O)cc3)c(Br)n(Cc3ccccc3)c2n1

nearest known ligand 0.63

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
DHFR P00374 13/20 0.52
TYMS P04818 6/20 0.52
GART P22102 2/20 0.47
ATIC P31939 2/20 0.47
FOLR2 P14207 1/20 0.47
FOLR1 P15328 1/20 0.47
SHMT1 P34896 1/20 0.47
SLC19A1 P41440 1/20 0.47
FRK P42685 1/20 0.47
SLC46A1 Q96NT5 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9844856 0.86 DHFR (0.43) DHFRTYMS
SCHEMBL9844852 0.86 DHFR (0.43) DHFRTYMS
Butane SCHEMBL9844926 0.86 DHFR (0.40) DHFRTYMSGARTATICFOLR2
SCHEMBL9844793 0.84 DHFR (0.55) DHFRTYMSGARTATICFOLR2
SCHEMBL9844802 0.84 AGTR1 (0.40)
Butane SCHEMBL9844893 0.81 DHFR (0.55) DHFRTYMSGARTATICFOLR2
SCHEMBL9556787 0.81 DRD2 (0.45)
SCHEMBL9844820 0.78 DHFR (0.61) DHFRTYMSGARTATICFOLR2
SCHEMBL9844817 0.78 DHFR (0.61) DHFRTYMSGARTATICFOLR2
SCHEMBL9339136 0.77 GART (0.68) DHFRTYMSGARTATICFOLR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0438261-A2 Condensed heterocyclic glutamic acid derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1991-07-24 EP claimed
EP-0438261-A2 Condensed heterocyclic glutamic acid derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1991-07-24 EP disclosed