SCHEMBL9846091

SCHEMBL9846091

Cc1nc(OCc2ccccc2)c(C#N)cc1C(N)=O

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.53
KDM4E B2RXH2 3/20 0.53
HPGD P15428 2/20 0.53
CRHBP P24387 2/20 0.53
CRHR2 Q13324 2/20 0.53
SMN1; SMN2 Q16637 3/20 0.52
HTT P42858 1/20 0.52
HSD17B10 Q99714 1/20 0.51
TDP1 Q9NUW8 1/20 0.48
POLB P06746 1/20 0.47
GAA P10253 1/20 0.47
XDH P47989 2/20 0.47
CNR1 P21554 1/20 0.47
HDAC1 Q13547 1/20 0.45
CYP1A2 P05177 2/20 0.44
CYP2C9 P11712 2/20 0.44
CYP2C19 P33261 2/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
LMNA P02545 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9585493 0.89 HTT (0.65) ALDH1A1KDM4EHPGDCRHBPCRHR2
SCHEMBL9846090 0.86 KDM4E (0.69) ALDH1A1KDM4EHPGDCRHBPCRHR2
SCHEMBL9846083 0.84 HTT (0.50) ALDH1A1KDM4EHPGDCRHBPCRHR2
SCHEMBL9846310 0.80 MEN1 (0.45) ALDH1A1KDM4ESMN1; SMN2HTTGAA
SCHEMBL23120426 0.77 CYP1A2 (0.51) ALDH1A1KDM4EHPGDCRHBPCRHR2
SCHEMBL23135737 0.77 CYP1A2 (0.58) ALDH1A1KDM4EHPGDCRHBPCRHR2
SCHEMBL9586720 0.77 ALDH1A1 (0.48) ALDH1A1KDM4EHPGDCRHBPCRHR2
SCHEMBL9846264 0.75 CNR1 (0.47) ALDH1A1KDM4EHPGDCRHBPCRHR2
SCHEMBL2624180 0.75 L3MBTL1 (0.60) KDM4EHPGDSMN1; SMN2HTTLMNA
SCHEMBL16616758 0.74 MCL1 (0.55) SMN1; SMN2HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0462800-A2 Inhibitors of HIV reverse transcriptase MERCK & CO. INC. (US) 1991-12-27 EP disclosed