SCHEMBL9846203

SCHEMBL9846203

CCc1cc(NCc2nc(CC)c(C)cc2OC)c(=O)[nH]c1C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 6/20 0.38
PDE3A Q14432 6/20 0.38
CRHR1 P34998 1/20 0.35
MAPT P10636 5/20 0.34
KDM4E B2RXH2 4/20 0.34
APAF1 O14727 1/20 0.34
RECQL P46063 1/20 0.34
GAA P10253 2/20 0.34
PDE10A Q9Y233 3/20 0.32
ALDH1A1 P00352 1/20 0.32
LMNA P02545 1/20 0.32
PLK4 O00444 1/20 0.32
CHEK1 O14757 1/20 0.32
AURKA O14965 1/20 0.32
NTRK1 P04629 1/20 0.32
LCK P06239 1/20 0.32
CDK1 P06493 1/20 0.32
CSF1R P07333 1/20 0.32
PIM1 P11309 1/20 0.32
RPS6KB1 P23443 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9846298 0.91 PDE3B (0.38) PDE3BPDE3ACRHR1MAPTKDM4E
SCHEMBL9682064 0.87 MAPT (0.34) CRHR1MAPTKDM4EAPAF1RECQL
SCHEMBL9846175 0.86 PDE3B (0.38) PDE3BPDE3AMAPTKDM4EAPAF1
SCHEMBL9168694 0.82 PDE3B (0.42) PDE3BPDE3AMAPTKDM4EAPAF1
SCHEMBL9846183 0.81 RXFP1 (0.38) PDE3BPDE3AMAPTKDM4EAPAF1
SCHEMBL9846165 0.81 PDE3B (0.41) PDE3BPDE3AMAPTKDM4EAPAF1
SCHEMBL9846246 0.78 MAPT (0.34) MAPTKDM4EAPAF1RECQLGAA
SCHEMBL9680359 0.78 MAPT (0.34) MAPTKDM4EAPAF1RECQLGAA
SCHEMBL9170296 0.76 KDM4E (0.44) PDE3BPDE3AMAPTKDM4EAPAF1
SCHEMBL9846107 0.75 PDE3B (0.41) PDE3BPDE3AMAPTKDM4EAPAF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0462800-A2 Inhibitors of HIV reverse transcriptase MERCK & CO. INC. (US) 1991-12-27 EP disclosed