SCHEMBL9847728

SCHEMBL9847728

NC(=O)Cc1nc2cc(F)c(N3CCCC3C(=O)O)cc2n1C1CC1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
OGFRL1 Q5TC84 5/20 0.38
KMT2A Q03164 1/20 0.37
CYP11B2 P19099 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.34
OPRM1 P35372 2/20 0.34
OPRK1 P41145 2/20 0.34
OPRD1 P41143 1/20 0.34
SPR P35270 1/20 0.34
OPRL1 P41146 2/20 0.34
CYP11B1 P15538 1/20 0.33
CPT1A P50416 1/20 0.33
ALK Q9UM73 3/20 0.33
ELANE P08246 2/20 0.33
JAK2 O60674 1/20 0.33
TYK2 P29597 1/20 0.33
JAK3 P52333 1/20 0.33
HPGD P15428 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9301733 0.80 CYP11B2 (0.40) CYP11B2SMN1; SMN2CYP11B1CPT1AJAK2
SCHEMBL9303690 0.74 OPRM1 (0.37) OGFRL1OPRM1OPRK1OPRD1CPT1A
SCHEMBL9301930 0.67 HTT (0.45) KMT2ACYP11B2SMN1; SMN2CYP11B1HPGD
SCHEMBL2935668 0.64 SMN1; SMN2 (0.42) KMT2ASMN1; SMN2
SCHEMBL9301581 0.63 HTT (0.50) OGFRL1KMT2ACYP11B2SMN1; SMN2OPRM1
SCHEMBL8140544 0.63 CCR1 (0.47) KMT2ASMN1; SMN2
SCHEMBL7548869 0.63 CCR1 (0.47) KMT2ASMN1; SMN2
SCHEMBL16759937 0.62 NOTUM (0.52) OGFRL1KMT2ASMN1; SMN2
SCHEMBL2034147 0.60 SMN1; SMN2 (0.46) OGFRL1KMT2ASMN1; SMN2HPGD
SCHEMBL21660807 0.59 HTT (0.43) KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0433648-A1 Substituted pyrimidobenzimidazole derivatives F. HOFFMANN-LA ROCHE AG (CH) 1991-06-26 EP disclosed