SCHEMBL9303690

SCHEMBL9303690

CC(C)(C)OC(=O)[C@@H]1CCCN1c1cc2c(cc1F)nc(CC(=O)NOCc1ccccc1)n2C1CC1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 3/20 0.37
OPRD1 P41143 3/20 0.37
OGFRL1 Q5TC84 3/20 0.37
OPRK1 P41145 2/20 0.37
ADORA3 P0DMS8 1/20 0.36
ADORA2A P29274 1/20 0.36
ADORA2B P29275 1/20 0.36
ADORA1 P30542 1/20 0.36
ACE P12821 2/20 0.35
RORC P51449 2/20 0.35
KLK7 P49862 1/20 0.35
AADAT Q8N5Z0 2/20 0.35
TRPV1 Q8NER1 1/20 0.35
ALK Q9UM73 3/20 0.34
CPT1A P50416 1/20 0.34
MET P08581 1/20 0.33
HDAC1 Q13547 2/20 0.32
HDAC8 Q9BY41 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
ATR Q13535 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9847716 0.85 HDAC1 (0.36) OPRM1OPRD1OGFRL1OPRK1RORC
SCHEMBL9301818 0.85 ATR (0.35) OPRM1OPRD1OGFRL1OPRK1RORC
SCHEMBL9302252 0.85 ACHE (0.42) OPRM1OPRD1OGFRL1RORC
SCHEMBL9302144 0.83 GRM5 (0.39) OPRM1OPRD1OGFRL1OPRK1CPT1A
SCHEMBL9303841 0.82 HPGD (0.35) OPRM1OPRD1OGFRL1OPRK1RORC
SCHEMBL9301969 0.81 GRM5 (0.42) OPRM1OPRD1OGFRL1OPRK1RORC
SCHEMBL9847728 0.74 OGFRL1 (0.38) OPRM1OPRD1OGFRL1OPRK1ALK
SCHEMBL9303648 0.72 ACE (0.34) OPRM1OPRD1OGFRL1OPRK1ADORA3
SCHEMBL9301682 0.71 RORC (0.42) OPRM1OPRD1OGFRL1RORC
SCHEMBL9303809 0.71 HTT (0.41) OPRM1OPRD1OGFRL1RORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5283248-A Bactericides, enzyme inhibitor of DNA-gyrase in bacteria HOFFMANN-LA ROCHE INC. (US) 1994-02-01 US disclosed
EP-0433648-A1 Substituted pyrimidobenzimidazole derivatives F. HOFFMANN-LA ROCHE AG (CH) 1991-06-26 EP disclosed