SCHEMBL9849202

SCHEMBL9849202

NC(=O)c1nccc2ccc(CCO[PH](=O)OCCc3ccc4ccnc(C(N)=O)c4c3)cc12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLAU P00749 5/20 0.40
HDAC1 Q13547 3/20 0.35
HDAC6 Q9UBN7 3/20 0.35
HDAC3 O15379 2/20 0.35
HDAC4 P56524 2/20 0.35
HDAC7 Q8WUI4 2/20 0.35
HDAC2 Q92769 2/20 0.35
HDAC10 Q969S8 2/20 0.35
HDAC11 Q96DB2 2/20 0.35
HDAC8 Q9BY41 2/20 0.35
HDAC9 Q9UKV0 2/20 0.35
HDAC5 Q9UQL6 2/20 0.35
CYP1A2 P05177 2/20 0.35
CYP2D6 P10635 2/20 0.35
CYP2C19 P33261 2/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
HIF1A Q16665 1/20 0.35
PLAT P00750 2/20 0.33
RAB9A P51151 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9849204 0.91 PLAU (0.40) PLAUHDAC1HDAC6HDAC3HDAC4
SCHEMBL9849459 0.77 PLAU (0.42) PLAUHDAC1HDAC6HDAC3HDAC4
SCHEMBL9849066 0.76 PLAU (0.33) PLAU
SCHEMBL9849320 0.75 PLAU (0.44) PLAUPLATAPAF1NSD2CASP3
SCHEMBL18526638 0.73 RAB9A (0.40) PLAUHDAC1HDAC6HDAC3HDAC4
SCHEMBL9849325 0.71 PLAU (0.43) PLAUHDAC1HDAC6HDAC3HDAC4
SCHEMBL9849065 0.69 PLAU (0.34) PLAU
SCHEMBL6027557 0.68 PLAU (0.64) PLAUPLATAPAF1NSD2CASP3
SCHEMBL16246728 0.67 PLAU (0.38) PLAUHDAC1HDAC6HDAC3HDAC4
SCHEMBL9849130 0.66 PLAU (0.38) PLAUHDAC1HDAC6HDAC3HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0421436-A2 Substituted carboxytetrahydroisoquinolines and derivatives thereof having pharmaceutical activity WARNER-LAMBERT COMPANY (US) 1991-04-10 EP disclosed