SCHEMBL9849404

SCHEMBL9849404

Nc1cc(CCCn2ccnc2)nc2cc(C(F)(F)F)ccc12

nearest known ligand 0.47

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 4/20 0.47
TBXAS1 P24557 2/20 0.43
HMOX1 P09601 1/20 0.41
CYP19A1 P11511 1/20 0.41
ATP4A P20648 1/20 0.41
ATP4B P51164 1/20 0.41
MCHR1 Q99705 3/20 0.40
QPCT Q16769 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9849430 0.82 TSHR (0.50) TBXAS1CYP19A1QPCT
SCHEMBL439523 0.75 MCHR1 (0.57) MCHR1
SCHEMBL9849409 0.72 NOS1 (0.50) NOS1QPCT
SCHEMBL9849597 0.69 SOD1 (0.48) CYP19A1QPCT
SCHEMBL10283707 0.68 NOS1 (0.67) NOS1TBXAS1HMOX1CYP19A1
Hydrochloric Acid SCHEMBL410883 0.67 NOS1 (0.65) NOS1TBXAS1HMOX1CYP19A1ATP4A
SCHEMBL437720 0.67 MCHR1 (0.69) MCHR1
SCHEMBL1264932 0.67 TBXAS1 (0.60) NOS1TBXAS1CYP19A1
SCHEMBL28803051 0.66 CYP19A1 (0.49) TBXAS1HMOX1CYP19A1
SCHEMBL3828474 0.66 BACE1 (0.45) MCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0446604-A2 Pyridine and related aza heterocycle derivatives as cardiovascular agents AMERICAN CYANAMID COMPANY (US) 1991-09-18 EP disclosed