SCHEMBL9849573

SCHEMBL9849573

Cc1c(CCCn2ccnc2)c(N)nc2c(C)cccc12

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.49
MEN1 O00255 3/20 0.49
LMNA P02545 3/20 0.47
TSHR P16473 3/20 0.47
ALDH1A1 P00352 3/20 0.47
HPGD P15428 2/20 0.47
MAPK1 P28482 2/20 0.47
ALOX15 P16050 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
KDM4E B2RXH2 1/20 0.44
POLB P06746 1/20 0.44
CASP1 P29466 1/20 0.44
CLK1 P49759 1/20 0.44
CASP7 P55210 1/20 0.44
HSD17B10 Q99714 1/20 0.44
PRKCI P41743 1/20 0.42
QPCT Q16769 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9849331 0.86 QPCT (0.45) KMT2AMEN1LMNATSHRALDH1A1
SCHEMBL9849295 0.83 TSHR (0.55) TSHRALDH1A1MAPK1ALOX15HSD17B10
SCHEMBL9849636 0.80 TSHR (0.54) TSHRALDH1A1MAPK1
SCHEMBL9849547 0.73 QPCT (0.50) KMT2AMEN1TSHRALDH1A1MAPK1
SCHEMBL9849881 0.72 GAA (0.55) KMT2AMEN1LMNATSHRALDH1A1
SCHEMBL20701924 0.72 PRKCI (0.53) KMT2AMEN1LMNATSHRALDH1A1
SCHEMBL9849578 0.71 ALDH1A1 (0.61) KMT2AMEN1LMNATSHRALDH1A1
SCHEMBL9849597 0.68 SOD1 (0.48) TSHRALDH1A1KDM4EPOLBQPCT
SCHEMBL9849395 0.68 CYP19A1 (0.52) TSHRALDH1A1MAPK1ALOX15POLB
SCHEMBL28803051 0.68 CYP19A1 (0.49) KMT2AMEN1PRKCI

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0446604-A2 Pyridine and related aza heterocycle derivatives as cardiovascular agents AMERICAN CYANAMID COMPANY (US) 1991-09-18 EP disclosed