SCHEMBL9850361

SCHEMBL9850361

COc1ccc(C(=O)C(O)c2ccccc2)c(N)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.44
CYP1A2 P05177 2/20 0.44
PGR P06401 2/20 0.44
HPGD P15428 2/20 0.44
SLC6A2 P23975 2/20 0.44
CYP2C19 P33261 2/20 0.44
ALDH1A1 P00352 2/20 0.44
CYP2D6 P10635 1/20 0.44
PDE4A P27815 1/20 0.44
MAPK1 P28482 1/20 0.44
HRH1 P35367 1/20 0.44
HTT P42858 1/20 0.44
SLC6A3 Q01959 1/20 0.44
PDE4D Q08499 1/20 0.44
CES2 O00748 1/20 0.44
CES1 P23141 1/20 0.44
L3MBTL1 Q9Y468 2/20 0.43
TDP1 Q9NUW8 2/20 0.43
AKR1C3 P42330 1/20 0.43
AKR1C2 P52895 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11283361 0.84 TDP1 (0.55) LMNAHPGDALDH1A1PDE4AHTT
SCHEMBL28062466 0.84 LMNA (0.46) LMNACYP1A2PGRHPGDSLC6A2
SCHEMBL11246241 0.83 CPS1 (0.50) LMNACYP1A2PGRHPGDSLC6A2
SCHEMBL9056011 0.81 MAPT (0.53) LMNAALDH1A1HTTL3MBTL1TDP1
SCHEMBL9559907 0.79 ALDH1A1 (0.49) LMNACYP1A2PGRHPGDSLC6A2
SCHEMBL11224343 0.78 LMNA (0.55) LMNAHPGDALDH1A1CYP2D6MAPK1
SCHEMBL22807498 0.78 POLB (0.47) LMNAHPGDALDH1A1MAPK1CES2
SCHEMBL27939668 0.78 CES2 (0.47) LMNAALDH1A1MAPK1CES2CES1
SCHEMBL9850347 0.78 ABL1 (0.47) LMNACYP1A2HPGDCYP2C19ALDH1A1
SCHEMBL17709653 0.77 ALDH1A1 (0.60) LMNAHPGDALDH1A1MAPK1CES2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105518001-A MODIFIED BET-PROTEIN-INHIBITING DIHYDROQUINOXALINONES AND DIHYDROPYRIDOPYRAZINONES Bayer Pharma AG 2016-04-20 CN disclosed
EP-0433112-A1 Modified gangliosides and the functional derivatives thereof FIDIA S.p.A. (IT) 1991-06-19 EP disclosed