SCHEMBL9850618

SCHEMBL9850618

Cc1ccc(C(=O)C(C)Cn2ccnc2)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 1/20 0.52
ADRA2B P18089 1/20 0.52
DRD3 P35462 1/20 0.52
SIGMAR1 Q99720 1/20 0.52
HRH3 Q9Y5N1 1/20 0.52
CYP1A2 P05177 1/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2D6 P10635 1/20 0.52
CYP2C9 P11712 1/20 0.52
CYP2C19 P33261 1/20 0.52
ALDH1A1 P00352 4/20 0.51
LMNA P02545 1/20 0.51
CYP19A1 P11511 3/20 0.49
CYP11B1 P15538 1/20 0.49
CYP11B2 P19099 1/20 0.49
CYP26A1 O43174 4/20 0.45
TDP1 Q9NUW8 1/20 0.43
NAMPT P43490 1/20 0.43
TBXAS1 P24557 1/20 0.43
QPCT Q16769 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9850632 0.87 LMNA (0.51) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL9850630 0.87 CYP19A1 (0.52) ALDH1A1LMNACYP19A1CYP26A1TBXAS1
SCHEMBL9850662 0.86 CHRM2 (0.54) CHRM2ADRA2BDRD3SIGMAR1HRH3
SCHEMBL9850574 0.85 SMN1; SMN2 (0.47) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL11144915 0.85 CYP19A1 (0.60) CYP1A2CYP3A4ALDH1A1CYP19A1TDP1
SCHEMBL9850634 0.85 L3MBTL1 (0.44) ALDH1A1CYP19A1CYP26A1TDP1TBXAS1
SCHEMBL9850426 0.85 CYP26A1 (0.61) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL9850547 0.84 TBXAS1 (0.49) CYP19A1TBXAS1
Hydrochloric Acid SCHEMBL9850522 0.83 CYP11B1 (0.43) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL11149385 0.82 CYP19A1 (0.53) ALDH1A1LMNACYP19A1CYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0423524-A2 Propiophenone derivatives and their preparation and pharmaceutical use MARUHO Co., Ltd. (JP) 1991-04-24 EP disclosed