SCHEMBL9850662

SCHEMBL9850662

CCc1ccc(C(=O)C(C)Cn2ccnc2)cc1

nearest known ligand 0.54

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 1/20 0.54
CYP2D6 P10635 1/20 0.54
ADRA2B P18089 1/20 0.54
ADRA2C P18825 1/20 0.54
CHRM3 P20309 1/20 0.54
DRD3 P35462 1/20 0.54
OPRD1 P41143 1/20 0.54
KCNH2 Q12809 1/20 0.54
SIGMAR1 Q99720 1/20 0.54
HRH3 Q9Y5N1 1/20 0.54
TBXAS1 P24557 10/20 0.49
CYP19A1 P11511 4/20 0.46
PDE4A P27815 1/20 0.45
PDE4B Q07343 1/20 0.45
PDE4C Q08493 1/20 0.45
PDE4D Q08499 1/20 0.45
QPCT Q16769 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9850547 0.90 TBXAS1 (0.49) TBXAS1CYP19A1
SCHEMBL9850618 0.86 CHRM2 (0.52) CHRM2CYP2D6ADRA2BDRD3SIGMAR1
SCHEMBL9850632 0.85 LMNA (0.51) CYP2D6CYP19A1
SCHEMBL9850630 0.85 CYP19A1 (0.52) TBXAS1CYP19A1
Hydrochloric Acid SCHEMBL9850390 0.84 TBXAS1 (0.47) TBXAS1CYP19A1PDE4APDE4BPDE4C
SCHEMBL9850440 0.84 CYP19A1 (0.50) TBXAS1CYP19A1
SCHEMBL11144915 0.83 CYP19A1 (0.60) TBXAS1CYP19A1
SCHEMBL9850574 0.83 SMN1; SMN2 (0.47) CYP2D6CYP19A1
SCHEMBL9850426 0.83 CYP26A1 (0.61) CYP2D6CYP19A1
SCHEMBL9850634 0.80 L3MBTL1 (0.44) TBXAS1CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0423524-A2 Propiophenone derivatives and their preparation and pharmaceutical use MARUHO Co., Ltd. (JP) 1991-04-24 EP disclosed