SCHEMBL9852082

SCHEMBL9852082

COc1cccc(CN2CCC(NC(=O)c3occ4ccccc34)CC2)c1

nearest known ligand 0.73

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 5/20 0.73
MCHR1 Q99705 6/20 0.64
SIGMAR1 Q99720 1/20 0.61
MAOB P27338 2/20 0.57
KCNH2 Q12809 1/20 0.57
CCR3 P51677 1/20 0.56
F10 P00742 1/20 0.55
ACHE P22303 1/20 0.54
CHRM2 P08172 1/20 0.54
CHRM1 P11229 1/20 0.54
CHRM3 P20309 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9727095 0.91 DRD4 (0.72) DRD4MCHR1SIGMAR1MAOBCCR3
SCHEMBL9727135 0.86 DRD4 (0.67) DRD4MCHR1SIGMAR1MAOB
SCHEMBL9852245 0.85 DRD4 (0.55) DRD4MCHR1SIGMAR1MAOBACHE
Dimethylamine SCHEMBL9852061 0.85 DRD4 (0.63) DRD4MCHR1SIGMAR1MAOB
SCHEMBL9727235 0.83 DRD4 (0.58) DRD4MCHR1SIGMAR1MAOBKCNH2
Iodide SCHEMBL9852255 0.82 DRD4 (0.60) DRD4MCHR1SIGMAR1MAOBKCNH2
SCHEMBL9727123 0.81 DRD4 (0.69) DRD4MCHR1SIGMAR1MAOB
SCHEMBL9727173 0.81 SIGMAR1 (0.57) DRD4MCHR1SIGMAR1MAOBACHE
SCHEMBL9852062 0.81 DRD4 (0.71) DRD4MCHR1SIGMAR1MAOBKCNH2
SCHEMBL9727149 0.81 DRD4 (0.58) DRD4MCHR1SIGMAR1MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0416581-A1 Substituted N-benzylpiperidine amides G.D. Searle & Co. (US) 1991-03-13 EP claimed