SCHEMBL9852110

SCHEMBL9852110

Nc1nc(-c2ncccn2)ns1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 2/20 0.55
ADORA1 P30542 2/20 0.55
ADORA3 P0DMS8 1/20 0.55
ADORA2B P29275 1/20 0.55
PI4KA P42356 2/20 0.37
PI4KB Q9UBF8 2/20 0.37
PIK3CD O00329 1/20 0.37
PIP5K1C O60331 1/20 0.37
PIK3CG P48736 1/20 0.37
HSP90AA1 P07900 1/20 0.36
ALOX15 P16050 2/20 0.34
RAB9A P51151 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
CYP19A1 P11511 7/20 0.32
KDM4E B2RXH2 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
NOS1 P29475 2/20 0.32
ALDH1A1 P00352 2/20 0.32
TSHR P16473 1/20 0.32
HSD17B10 Q99714 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6003356 0.83 ADORA3 (0.58) ADORA2AADORA1ADORA3ADORA2BALOX15
SCHEMBL11273216 0.79 ADORA3 (0.48) ADORA2AADORA1ADORA3ADORA2BPI4KA
SCHEMBL3674565 0.78 KDM4E (0.56) ADORA2AADORA1ADORA3ADORA2BPI4KA
SCHEMBL30585765 0.78 KDM4E (0.56) ADORA2AADORA1ADORA3ADORA2BPI4KA
SCHEMBL20422809 0.75 ADORA3 (0.49) ADORA2AADORA1ADORA3ADORA2BRAB9A
SCHEMBL18377816 0.74 ADORA3 (0.47) ADORA2AADORA1ADORA3ADORA2BRAB9A
SCHEMBL16718760 0.74 ADORA3 (0.47) ADORA2AADORA1ADORA3ADORA2BPI4KA
SCHEMBL6529431 0.73 PSMD14 (0.30)
SCHEMBL69810 0.71 ADORA3 (1.00) ADORA2AADORA1ADORA3ADORA2BALOX15
SCHEMBL10391988 0.71 ADORA2A (0.49) ADORA2AADORA1ADORA3ADORA2BHSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0455356-A1 Substituted 5-amino-1,2,4-thiadiazoles with pharmaceutical activity LILLY INDUSTRIES LIMITED (GB) 1991-11-06 EP disclosed