SCHEMBL9857352

SCHEMBL9857352

NC(=O)c1nnn(Cc2ccc(F)cc2F)c1C(N)=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.43
MAPT P10636 3/20 0.41
KDM4E B2RXH2 4/20 0.40
ADORA3 P0DMS8 1/20 0.40
ADORA2A P29274 1/20 0.40
ADORA2B P29275 1/20 0.40
ADORA1 P30542 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
HDAC1 Q13547 1/20 0.40
KCNK3 O14649 3/20 0.40
AURKA O14965 1/20 0.38
RPS6KB1 P23443 1/20 0.38
AURKB Q96GD4 1/20 0.38
POLB P06746 1/20 0.38
MEN1 O00255 1/20 0.38
TRPA1 O75762 1/20 0.38
HPGD P15428 1/20 0.38
KMT2A Q03164 1/20 0.38
HSD17B10 Q99714 1/20 0.38
MAPK8 P45983 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9857331 0.90 TP53 (0.41) TP53MAPTADORA3ADORA2AADORA2B
SCHEMBL9857450 0.84 GRM2 (0.45) MAPTADORA3ADORA2AADORA2BADORA1
SCHEMBL10666237 0.83 NPC1 (0.48) TP53MAPTKDM4ESMN1; SMN2HDAC1
SCHEMBL9857464 0.79 CA5A (0.44) TP53MAPTKDM4EADORA3ADORA2A
SCHEMBL9857412 0.78 CA5A (0.55) TP53KDM4EADORA3ADORA2AADORA2B
SCHEMBL9857903 0.75 CA5A (0.46) MAPTKDM4EMEN1KMT2AHSD17B10
SCHEMBL9857974 0.73 LMNA (0.49) TP53MAPTSMN1; SMN2POLBMEN1
SCHEMBL18320969 0.73 PTGDR2 (0.38) TP53MAPTKDM4EADORA3ADORA2A
SCHEMBL9857419 0.72 CA5A (0.61) TP53MAPTKDM4ESMN1; SMN2HDAC1
SCHEMBL10665851 0.72 NPC1 (0.48) TP53ADORA3ADORA2AADORA2BADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0199262-B1 FLUORINATED BENZYL TRIAZOLE COMPOUNDS CIBA-GEIGY AG (CH) 1991-02-27 EP claimed
EP-0199262-A2 Fluorinated benzyl triazole compounds CIBA-GEIGY AG (CH) 1986-10-29 EP claimed
EP-0199262-B1 FLUORINATED BENZYL TRIAZOLE COMPOUNDS CIBA-GEIGY AG (CH) 1991-02-27 EP disclosed
US-4789680-A Aralkyltriazole compounds CIBA-GEIGY CORPORATION (US) 1988-12-06 US disclosed
EP-0199262-A2 Fluorinated benzyl triazole compounds CIBA-GEIGY AG (CH) 1986-10-29 EP disclosed