SCHEMBL9857331

SCHEMBL9857331

NC(=O)c1nnn(Cc2cc(F)ccc2F)c1C(N)=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.41
ADORA3 P0DMS8 1/20 0.40
ADORA2A P29274 1/20 0.40
ADORA2B P29275 1/20 0.40
ADORA1 P30542 1/20 0.40
ROCK2 O75116 2/20 0.39
TSHR P16473 1/20 0.39
RORC P51449 3/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
MAPT P10636 1/20 0.38
MAPK8 P45983 1/20 0.38
DPP4 P27487 1/20 0.37
GALR3 O60755 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37
NR2F2 P24468 1/20 0.37
HIF1A Q16665 1/20 0.37
KCNMA1 Q12791 1/20 0.37
CA5A P35218 1/20 0.36
PTGDR2 Q9Y5Y4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9857352 0.90 TP53 (0.43) TP53ADORA3ADORA2AADORA2BADORA1
SCHEMBL9857450 0.84 GRM2 (0.45) ADORA3ADORA2AADORA2BADORA1TSHR
SCHEMBL10665851 0.83 NPC1 (0.48) TP53ADORA3ADORA2AADORA2BADORA1
SCHEMBL9857464 0.79 CA5A (0.44) TP53ADORA3ADORA2AADORA2BADORA1
SCHEMBL9857412 0.78 CA5A (0.55) TP53ADORA3ADORA2AADORA2BADORA1
SCHEMBL9857974 0.73 LMNA (0.49) TP53TSHRSMN1; SMN2MAPTGALR3
SCHEMBL9857903 0.73 CA5A (0.46) TSHRMAPTCA5A
SCHEMBL10666237 0.72 NPC1 (0.48) TP53SMN1; SMN2MAPTPTGDR2
SCHEMBL9858313 0.72 CA5A (0.61) MAPTMAPK8DPP4CA5ARIPK1
SCHEMBL9634851 0.72 HPGD (0.61) TSHRSMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0199262-B1 FLUORINATED BENZYL TRIAZOLE COMPOUNDS CIBA-GEIGY AG (CH) 1991-02-27 EP claimed
US-4789680-A Aralkyltriazole compounds CIBA-GEIGY CORPORATION (US) 1988-12-06 US claimed
EP-0199262-A2 Fluorinated benzyl triazole compounds CIBA-GEIGY AG (CH) 1986-10-29 EP claimed
EP-0199262-B1 FLUORINATED BENZYL TRIAZOLE COMPOUNDS CIBA-GEIGY AG (CH) 1991-02-27 EP disclosed
US-4789680-A Aralkyltriazole compounds CIBA-GEIGY CORPORATION (US) 1988-12-06 US disclosed
EP-0199262-A2 Fluorinated benzyl triazole compounds CIBA-GEIGY AG (CH) 1986-10-29 EP disclosed