SCHEMBL9857464

SCHEMBL9857464

NC(=O)c1nnn(Cc2cccc(F)c2F)c1C(N)=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA5A P35218 1/20 0.44
ADORA3 P0DMS8 1/20 0.42
ADORA2A P29274 1/20 0.42
ADORA2B P29275 1/20 0.42
ADORA1 P30542 1/20 0.42
AURKA O14965 1/20 0.39
PDPK1 O15530 1/20 0.39
RPS6KB1 P23443 1/20 0.39
GRM2 Q14416 1/20 0.38
RORC P51449 2/20 0.37
ALDH1A1 P00352 1/20 0.36
HTT P42858 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
PKM P14618 1/20 0.35
PKLR P30613 1/20 0.35
HPGD P15428 1/20 0.35
P2RX7 Q99572 2/20 0.34
TP53 P04637 1/20 0.34
MAPT P10636 1/20 0.34
PIK3CD O00329 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9857450 0.89 GRM2 (0.45) CA5AADORA3ADORA2AADORA2BADORA1
SCHEMBL9857412 0.86 CA5A (0.55) CA5AADORA3ADORA2AADORA2BADORA1
SCHEMBL9857903 0.81 CA5A (0.46) CA5AALDH1A1MAPTKDM4E
SCHEMBL9857331 0.79 TP53 (0.41) CA5AADORA3ADORA2AADORA2BADORA1
SCHEMBL9857352 0.79 TP53 (0.43) ADORA3ADORA2AADORA2BADORA1AURKA
SCHEMBL10664842 0.79 TP53 (0.54) ALDH1A1HTTNPSR1TP53
SCHEMBL9857974 0.78 LMNA (0.49) ALDH1A1NPSR1HPGDTP53MAPT
SCHEMBL9475577 0.76 HPGD (0.52) ADORA3ADORA2AADORA2BADORA1GRM2
SCHEMBL10662709 0.75 CA5A (0.49) CA5AADORA3ADORA2AADORA2BADORA1
SCHEMBL9634851 0.75 HPGD (0.61) ALDH1A1HTTHPGDMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0199262-B1 FLUORINATED BENZYL TRIAZOLE COMPOUNDS CIBA-GEIGY AG (CH) 1991-02-27 EP claimed
EP-0199262-A2 Fluorinated benzyl triazole compounds CIBA-GEIGY AG (CH) 1986-10-29 EP claimed
EP-0199262-B1 FLUORINATED BENZYL TRIAZOLE COMPOUNDS CIBA-GEIGY AG (CH) 1991-02-27 EP disclosed
US-4789680-A Aralkyltriazole compounds CIBA-GEIGY CORPORATION (US) 1988-12-06 US disclosed
EP-0199262-A2 Fluorinated benzyl triazole compounds CIBA-GEIGY AG (CH) 1986-10-29 EP disclosed