SCHEMBL985879

SCHEMBL985879

COc1ccc(-c2ncnc3c(C(=O)NC4CCN(C(=O)C5CC5)CC4)c[nH]c23)c(OCC2CC2)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1B P49286 1/20 0.40
PAK1 Q13153 1/20 0.38
HPGDS O60760 1/20 0.38
HTR4 Q13639 1/20 0.37
TSHR P16473 1/20 0.37
TLR9 Q9NR96 1/20 0.36
TLR7 Q9NYK1 1/20 0.36
MDM4 O15151 1/20 0.36
PRKAB2 O43741 2/20 0.35
PRKAG1 P54619 2/20 0.35
PRKAA2 P54646 2/20 0.35
PRKAA1 Q13131 2/20 0.35
PRKAG3 Q9UGI9 2/20 0.35
PRKAG2 Q9UGJ0 2/20 0.35
PRKAB1 Q9Y478 2/20 0.35
MCHR1 Q99705 2/20 0.35
JAK1 P23458 1/20 0.35
JAK3 P52333 1/20 0.35
CYP4F2 P78329 1/20 0.35
CYP4A11 Q02928 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL981830 0.94 MTNR1B (0.40) MTNR1BPAK1HPGDSHTR4TSHR
SCHEMBL984587 0.93 HPGDS (0.44) PAK1HPGDSHTR4TSHRMDM4
SCHEMBL982565 0.92 HPGDS (0.39) MTNR1BPAK1HPGDSHTR4TSHR
SCHEMBL984353 0.91 TBK1 (0.41) PAK1HPGDSHTR4TSHRMDM4
SCHEMBL983581 0.91 BTK (0.40) PAK1HPGDSHTR4TSHRMDM4
SCHEMBL983426 0.91 ALDH1A1 (0.44)
SCHEMBL985429 0.90 PAK1 (0.38) PAK1HPGDSHTR4TSHRMDM4
SCHEMBL984925 0.89 HTR4 (0.39) MTNR1BHPGDSHTR4GRIN1GRIN2B
SCHEMBL983065 0.89 HTR4 (0.39) MTNR1BHPGDSHTR4GRIN1GRIN2B
SCHEMBL984605 0.89 HTR4 (0.39) MTNR1BHPGDSHTR4GRIN1GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110021479-A1 PYRROLOPYRIMIDINECARBOXAMIDES NYCOMED GMBH (DE) 2011-01-27 US claimed
US-20110021479-A1 PYRROLOPYRIMIDINECARBOXAMIDES NYCOMED GMBH (DE) 2011-01-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110021479-A1 PYRROLOPYRIMIDINECARBOXAMIDES PDE5A, PDE3A, PDE2A MTNR1B 2849/4885PAK1 1999/4885HPGDS 651/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.