SCHEMBL9859266

SCHEMBL9859266

O=C=Nc1ccc(Br)c(Cl)c1OC(F)F

nearest known ligand 0.32

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.32
ALDH1A1 P00352 1/20 0.32
HPGD P15428 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
ALOX15 P16050 1/20 0.32
GFER P55789 1/20 0.32
ADAM17 P78536 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11082116 0.86 TDP1 (0.36) CYP3A4ALDH1A1HPGDTDP1
SCHEMBL11535245 0.83 TDP1 (0.34) CYP3A4ALDH1A1HPGDTDP1
SCHEMBL9859078 0.80 CYP3A4 (0.32) CYP3A4ALDH1A1HPGDTDP1
SCHEMBL9859297 0.79 CYP3A4 (0.42) CYP3A4
SCHEMBL11473361 0.79 TDP1 (0.36) CYP3A4ALDH1A1HPGDTDP1
SCHEMBL11531900 0.76 CYP3A4 (0.42) CYP3A4ALDH1A1TDP1
SCHEMBL11471789 0.70 CYP3A4 (0.42) CYP3A4ALDH1A1HPGDTDP1
SCHEMBL9859146 0.70 CYP3A4 (0.42) CYP3A4ALDH1A1HPGDTDP1
SCHEMBL21239547 0.68 ALOX15 (0.40) CYP3A4ALDH1A1HPGDTDP1ALOX15
SCHEMBL29874044 0.68 ALOX15 (0.40) CYP3A4ALDH1A1HPGDTDP1ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0153127-B1 N-ARYL-3-ARYL-4,5-DIHYDRO-1H-PYRAZOLE-1-CARBOXAMIDES, PROCESSES FOR THEIR PRODUCTION, INSECTICIDAL COMPOSITIONS CONTAINING THEM AND METHODS FOR COMBATTING INSECTS ROHM AND HAAS COMPANY (US) 1991-04-03 EP disclosed
US-4863947-A PESTICIDES, INSECTICIDES ROHM AND HAAS (US) 1989-09-05 US disclosed
US-4663341-A Insecticidal n-aryl-3-aryl-4,5-dihydro-1h-pyrazole-1-carboxamides ROHM AND HAAS COMPANY (US) 1987-05-05 US disclosed
EP-0153127-A2 N-aryl-3-aryl-4,5-dihydro-1H-pyrazole-1-carboxamides, processes for their production, insecticidal compositions containing them and methods for combatting insects ROHM AND HAAS COMPANY (US) 1985-08-28 EP disclosed