SCHEMBL9859767

SCHEMBL9859767

CN(C)C(=O)CC(=O)c1ccc(C(F)(F)F)c(Cl)c1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 1/20 0.42
XPO1 O14980 1/20 0.40
CCR2 P41597 5/20 0.39
RAPGEF3 O95398 2/20 0.38
NOTUM Q6P988 2/20 0.38
MEN1 O00255 1/20 0.38
ALDH1A1 P00352 1/20 0.38
KMT2A Q03164 1/20 0.38
MRGPRX4 Q96LA9 1/20 0.38
KCNH2 Q12809 1/20 0.38
POLQ O75417 1/20 0.37
KDR P35968 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C19 P33261 1/20 0.37
RAB9A P51151 1/20 0.37
HTT P42858 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9859293 0.81 MEN1 (0.47) GPBAR1RAPGEF3NOTUMMEN1KMT2A
SCHEMBL24959794 0.80 NOTUM (0.42) GPBAR1RAPGEF3NOTUMALDH1A1MRGPRX4
SCHEMBL9858842 0.79 HDAC1 (0.47) GPBAR1RAPGEF3NOTUMMRGPRX4KDR
SCHEMBL25403646 0.78 PLOD2 (0.41) GPBAR1RAPGEF3NOTUMMEN1ALDH1A1
SCHEMBL23112384 0.77 GSK3B (0.54) NOTUMMRGPRX4
SCHEMBL313146 0.75 KIF11 (0.54) GPBAR1RAPGEF3NOTUMMRGPRX4KDR
SCHEMBL6578591 0.74 ALDH1A1 (0.50) ALDH1A1MRGPRX4KDRCYP1A2CYP2D6
SCHEMBL28144725 0.74 NOTUM (0.67) NOTUMMEN1ALDH1A1KMT2AMRGPRX4
SCHEMBL9481842 0.74 NPC1 (0.47) MEN1ALDH1A1KMT2ARAB9A
SCHEMBL665618 0.74 CA12 (0.51) NOTUMALDH1A1CYP1A2RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0153127-B1 N-ARYL-3-ARYL-4,5-DIHYDRO-1H-PYRAZOLE-1-CARBOXAMIDES, PROCESSES FOR THEIR PRODUCTION, INSECTICIDAL COMPOSITIONS CONTAINING THEM AND METHODS FOR COMBATTING INSECTS ROHM AND HAAS COMPANY (US) 1991-04-03 EP disclosed
US-4863947-A PESTICIDES, INSECTICIDES ROHM AND HAAS (US) 1989-09-05 US disclosed
US-4663341-A Insecticidal n-aryl-3-aryl-4,5-dihydro-1h-pyrazole-1-carboxamides ROHM AND HAAS COMPANY (US) 1987-05-05 US disclosed
EP-0153127-A2 N-aryl-3-aryl-4,5-dihydro-1H-pyrazole-1-carboxamides, processes for their production, insecticidal compositions containing them and methods for combatting insects ROHM AND HAAS COMPANY (US) 1985-08-28 EP disclosed