SCHEMBL9861341

SCHEMBL9861341

Nc1c(Cc2ccccc2)cc(C(F)(F)F)c2ccccc12

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.45
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
KDM4E B2RXH2 1/20 0.41
LMNA P02545 1/20 0.41
MAPT P10636 1/20 0.41
MAPK1 P28482 1/20 0.41
HTT P42858 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
LIMK1 P53667 1/20 0.39
LTA4H P09960 1/20 0.38
BCL2 P10415 1/20 0.38
BCL2L1 Q07817 1/20 0.38
NR1H2 P55055 4/20 0.37
NR1H3 Q13133 4/20 0.37
HTR2A P28223 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9861413 0.81 BCL2 (0.46) BCL2BCL2L1
SCHEMBL9861455 0.80 KDM4E (0.44) BACE1MEN1KMT2AKDM4ELMNA
SCHEMBL9861521 0.75 LTA4H (0.47) KDM4ELIMK1LTA4HHTR2A
SCHEMBL6198894 0.73 GAA (0.48) BACE1KDM4EMAPTLIMK1LTA4H
SCHEMBL5380250 0.71 KDM4E (0.56) KDM4ENPSR1LTA4HBCL2BCL2L1
SCHEMBL9861294 0.71 TACR1 (0.39) LIMK1BCL2BCL2L1HTR2A
SCHEMBL24332883 0.70 KDM4E (0.47) BACE1MEN1KMT2AKDM4ELMNA
SCHEMBL9861395 0.70 KMT2A (0.47) BACE1MEN1KMT2AKDM4ELMNA
SCHEMBL9861634 0.69 KDM4E (0.54) BACE1MEN1KMT2AKDM4ELMNA
SCHEMBL28492984 0.69 CALM1 (0.55) MEN1KMT2ABCL2BCL2L1HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5008425-A Trifluoromethylation of carbonyl compounds ETHYL CORPORATION (US) 1991-04-16 US disclosed
EP-0336371-A2 Gem-disubstituted cyclohexadienones and their production ETHYL CORPORATION (US) 1989-10-11 EP disclosed
US-4871877-A Gem-disubstituted cyclohexadienones and their production ETHYL CORPORATION (US) 1989-10-03 US disclosed
US-4845258-A Production of gem-disubstituted cyclohexadienones ETHYL CORPORATION (US) 1989-07-04 US disclosed
US-4804774-A Production of gem-disubstituted cyclohexadienones ETHYL CORPORATION (US) 1989-02-14 US disclosed
US-4804772-A Gem-disubstituted cyclohexadienones and their production ETHYL CORPORATION (US) 1989-02-14 US disclosed
US-4804773-A Production of gem-disubstituted cyclohexadienones ETHYL CORPORATION (US) 1989-02-14 US disclosed