SCHEMBL9864129

SCHEMBL9864129

CCC(O)C(N(C)CCN1CCOCC1)C1(c2cccc(C(F)(F)F)c2)CCC1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASR P41180 1/20 0.41
OPRM1 P35372 5/20 0.40
OPRL1 P41146 5/20 0.40
OPRD1 P41143 1/20 0.39
LMNA P02545 1/20 0.39
TACR1 P25103 1/20 0.38
TACR3 P29371 1/20 0.38
SLC6A2 P23975 2/20 0.38
SLC6A3 Q01959 2/20 0.38
SLC6A4 P31645 1/20 0.38
KDM4E B2RXH2 3/20 0.38
TRPV4 Q9HBA0 2/20 0.38
ALDH1A1 P00352 2/20 0.38
TDP1 Q9NUW8 1/20 0.38
GAA P10253 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
KMT2A Q03164 1/20 0.37
OPRK1 P41145 2/20 0.36
EPHX2 P34913 1/20 0.36
HTR2A P28223 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9864332 0.83 CASR (0.44) CASROPRM1OPRL1OPRD1LMNA
SCHEMBL9864359 0.80 SLC6A4 (0.48) OPRM1OPRL1OPRD1SLC6A2SLC6A3
SCHEMBL9863909 0.72 SLC6A4 (0.46) OPRM1OPRL1OPRD1SLC6A2SLC6A3
Hydrochloric Acid SCHEMBL9864247 0.72 SLC6A4 (0.46) OPRM1OPRL1OPRD1SLC6A2SLC6A3
SCHEMBL10637961 0.67 OPRM1 (0.36) OPRM1OPRL1OPRD1SLC6A2SLC6A3
SCHEMBL9118387 0.66 SLC6A4 (0.52) OPRM1OPRL1SLC6A2SLC6A3SLC6A4
SCHEMBL9864288 0.65 SLC6A4 (0.47) OPRM1OPRL1SLC6A2SLC6A3SLC6A4
SCHEMBL9864259 0.64 CHRM2 (0.45) TACR3SLC6A2SLC6A3SLC6A4KCNH2
SCHEMBL9864273 0.64 SLC6A4 (0.46) OPRM1OPRL1SLC6A2SLC6A3SLC6A4
Hydrochloric Acid SCHEMBL1521 0.62 SLC6A4 (0.48) OPRM1OPRL1OPRD1SLC6A2SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5047432-A Antidepressants THE BOOTS COMPANY PLC (GB) 1991-09-10 US disclosed
US-4925879-A ANTIDEPRESSANTS BOOTS COMPANY, PLC (GB) 1990-05-15 US disclosed
EP-0191542-B1 ARYLCYCLOBUTYLALKYL AMINES AND THEIR USE AS ANTIDEPRESSIVE MEDICINES The Boots Company PLC (GB) 1988-06-08 EP disclosed
EP-0191542-A1 Arylcyclobutylalkyl amines and their use as antidepressive medicines The Boots Company PLC (GB) 1986-08-20 EP disclosed