SCHEMBL9864633

SCHEMBL9864633

Cc1cccc2c(Cl)c(CCCl)nnc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.35
HTR1A P08908 1/20 0.34
ADRA1D P25100 1/20 0.34
ADRA1A P35348 1/20 0.34
ADRA1B P35368 1/20 0.34
CYP1A2 P05177 1/20 0.33
CYP2A6 P11509 1/20 0.33
KDM4E B2RXH2 4/20 0.33
HSP90AB1 P08238 1/20 0.33
HPGD P15428 4/20 0.32
TSHR P16473 3/20 0.32
HSD17B10 Q99714 2/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
PARP2 Q9UGN5 2/20 0.32
POLB P06746 1/20 0.32
TNKS O95271 1/20 0.32
TNKS2 Q9H2K2 1/20 0.32
RECQL P46063 1/20 0.32
RAD52 P43351 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24507816 0.75 CYP2A6 (0.41) ALDH1A1HTR1AADRA1DADRA1AADRA1B
SCHEMBL2830264 0.74 ALDH1A1 (0.58) ALDH1A1KDM4EHSP90AB1MEN1KMT2A
SCHEMBL9864036 0.73 GPR3 (0.46) ALDH1A1CYP1A2KDM4EHPGDKMT2A
SCHEMBL3279694 0.69 KDM4E (0.41) ALDH1A1CYP1A2KDM4EHPGDTSHR
SCHEMBL18436374 0.65 AXL (0.46) HTR1AADRA1DADRA1AADRA1BCYP1A2
SCHEMBL10810254 0.65 ELANE (0.44) ALDH1A1CYP1A2CYP2A6KDM4EHPGD
SCHEMBL11210067 0.64 CYP2A6 (0.41) ALDH1A1CYP1A2CYP2A6KDM4ETSHR
SCHEMBL2125784 0.63 KDM4E (0.49) ALDH1A1CYP1A2CYP2A6KDM4ETSHR
SCHEMBL10757356 0.63 CYP2A6 (0.39) ALDH1A1HTR1AADRA1DADRA1AADRA1B
SCHEMBL9865079 0.62 AR (0.44) CYP1A2KDM4EHPGDTSHRPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4988695-A Gastrointestinal disorders, antisecretory agents SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1991-01-29 US disclosed
EP-0380257-A2 Condensed cinnoline derivatives, process and intermediates for their preparation and pharmaceutical compositions containing them SMITHKLINE BECKMAN INTERCREDIT B.V. (NL) 1990-08-01 EP disclosed