SCHEMBL9865154

SCHEMBL9865154

CCNC1CC2CCC(C1)N2c1c(C(=O)O)c(=O)c2c(N)c(F)cc(F)c2n1C1CC1

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
FOXO1 Q12778 1/20 0.35
GSK3B P49841 12/20 0.35
TOP2A P11388 1/20 0.33
TOP2B Q02880 1/20 0.33
CACNA1F O60840 1/20 0.32
POLB P06746 1/20 0.32
MAPK1 P28482 1/20 0.32
CACNA1D Q01668 1/20 0.32
KCNH2 Q12809 1/20 0.32
CACNA1S Q13698 1/20 0.32
CACNA1C Q13936 1/20 0.32
CHRM1 P11229 3/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9866818 0.90 GSK3B (0.38) FOXO1GSK3BTOP2ATOP2BCACNA1F
SCHEMBL9865852 0.79 CHRM1 (0.34) CHRM1
SCHEMBL9866155 0.67 KDM4E (0.36) GSK3BTOP2ATOP2BPOLBCHRM1
SCHEMBL4716155 0.65 GSK3B (0.59) GSK3BTOP2ATOP2BCACNA1FPOLB
SCHEMBL9865560 0.64 TOP2A (0.54) GSK3BTOP2ATOP2BPOLBKCNH2
SCHEMBL3134076 0.64 KCNH2 (0.38) GSK3BTOP2ATOP2BPOLBKCNH2
SCHEMBL9865549 0.62 KDM4E (0.63) TOP2ATOP2B
SCHEMBL9865008 0.61 DPP4 (0.53) TOP2ATOP2BKCNH2
SCHEMBL9244385 0.61 KCNH2 (0.41) GSK3BPOLBKCNH2CHRM1
SCHEMBL4713790 0.61 TOP2A (0.61) GSK3BTOP2ATOP2BCACNA1FPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4992546-A Process for preparing 6,8-diazabicyclo[3.2.2]nonane derivatives WARNER-LAMBERT COMPANY (US) 1991-02-12 US disclosed
US-4968799-A Antibacterial agents WARNER-LAMBERT COMPANY (US) 1990-11-06 US disclosed
US-4962108-A A QUIN-4-ONE HAVING THE FOLLOWING RING SUBSTITUENTS; 1-ALKYL OR PHENYL, 3-CARBOXY DERIVATIVE, 6-FLUORO AND 8-BRIDGED N-HETEROCYCLIC RING WARNER-LAMBERT COMPANY (US) 1990-10-09 US disclosed
US-4923879-A CARBOXYLIC ACID DERIVATIVES WITH BRIDGED SIDECHAINS WARNER-LAMBERT COMPANY (US) 1990-05-08 US disclosed
EP-0305744-A2 Quinoline, naphthyridine and benzoxazine-carboxylic acid derivatives and their use as antibacterial agents WARNER-LAMBERT COMPANY (US) 1989-03-08 EP disclosed