SCHEMBL9866155

SCHEMBL9866155

CNC1CC2CCC(C1)N2c1c(C(=O)O)c(=O)c2cc(F)cc(Cl)c2n1C1CC1

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
CYP1A2 P05177 1/20 0.36
ALDH1A1 P00352 1/20 0.31
POLB P06746 1/20 0.31
CHRM2 P08172 1/20 0.31
CHRM1 P11229 1/20 0.31
OPRM1 P35372 1/20 0.31
OPRD1 P41143 1/20 0.31
CCR3 P51677 2/20 0.31
MAPT P10636 1/20 0.31
TOP2A P11388 2/20 0.31
TOP2B Q02880 2/20 0.31
P2RX7 Q99572 1/20 0.30
PIM1 P11309 1/20 0.30
GSK3A P49840 1/20 0.30
GSK3B P49841 1/20 0.30
PIM3 Q86V86 1/20 0.30
CSNK1G1 Q9HCP0 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9865852 0.89 CHRM1 (0.34) KDM4ESMN1; SMN2CYP1A2CHRM1CCR3
SCHEMBL9866818 0.77 GSK3B (0.38) POLBTOP2ATOP2BGSK3B
Hydrochloric Acid SCHEMBL6005743 0.74 ALDH1A1 (0.48) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL3315232 0.73 ALDH1A1 (0.43) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL4715010 0.68 KDM4E (0.57) KDM4ESMN1; SMN2CYP1A2ALDH1A1POLB
SCHEMBL9865154 0.67 FOXO1 (0.35) POLBCHRM1TOP2ATOP2BGSK3B
SCHEMBL8324882 0.67 CHRM2 (0.42) KDM4ECHRM2
SCHEMBL15134878 0.66 PDE2A (0.36) KDM4ESMN1; SMN2CYP1A2ALDH1A1POLB
SCHEMBL9249913 0.66 KCNH2 (0.41) KDM4ESMN1; SMN2CYP1A2ALDH1A1POLB
Heptane SCHEMBL8861899 0.64 KDM4E (0.52) KDM4ESMN1; SMN2CYP1A2ALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4992546-A Process for preparing 6,8-diazabicyclo[3.2.2]nonane derivatives WARNER-LAMBERT COMPANY (US) 1991-02-12 US disclosed
US-4968799-A Antibacterial agents WARNER-LAMBERT COMPANY (US) 1990-11-06 US disclosed
US-4962108-A A QUIN-4-ONE HAVING THE FOLLOWING RING SUBSTITUENTS; 1-ALKYL OR PHENYL, 3-CARBOXY DERIVATIVE, 6-FLUORO AND 8-BRIDGED N-HETEROCYCLIC RING WARNER-LAMBERT COMPANY (US) 1990-10-09 US disclosed
US-4923879-A CARBOXYLIC ACID DERIVATIVES WITH BRIDGED SIDECHAINS WARNER-LAMBERT COMPANY (US) 1990-05-08 US disclosed
EP-0305744-A2 Quinoline, naphthyridine and benzoxazine-carboxylic acid derivatives and their use as antibacterial agents WARNER-LAMBERT COMPANY (US) 1989-03-08 EP disclosed