SCHEMBL9866818

SCHEMBL9866818

CNC1CC2CCC(C1)N2c1c(C(=O)O)c(=O)c2c(N)c(F)cc(F)c2n1C1CC1

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 15/20 0.38
TOP2A P11388 2/20 0.36
TOP2B Q02880 2/20 0.36
CACNA1F O60840 1/20 0.35
POLB P06746 1/20 0.35
MAPK1 P28482 1/20 0.35
CACNA1D Q01668 1/20 0.35
KCNH2 Q12809 1/20 0.35
CACNA1S Q13698 1/20 0.35
CACNA1C Q13936 1/20 0.35
FOXO1 Q12778 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9865154 0.90 FOXO1 (0.35) GSK3BTOP2ATOP2BCACNA1FPOLB
SCHEMBL9866155 0.77 KDM4E (0.36) GSK3BTOP2ATOP2BPOLB
SCHEMBL4716155 0.69 GSK3B (0.59) GSK3BTOP2ATOP2BCACNA1FPOLB
SCHEMBL9865852 0.67 CHRM1 (0.34)
SCHEMBL4713790 0.65 TOP2A (0.61) GSK3BTOP2ATOP2BCACNA1FPOLB
SCHEMBL4673155 0.63 TOP2A (0.44) GSK3BTOP2ATOP2BCACNA1FPOLB
SCHEMBL4673154 0.63 TOP2A (0.44) GSK3BTOP2ATOP2BCACNA1FPOLB
SCHEMBL4719276 0.63 GSK3B (0.56) GSK3BTOP2ATOP2BCACNA1FPOLB
SCHEMBL6786216 0.62 GSK3B (0.40) GSK3BTOP2ATOP2BCACNA1FPOLB
SCHEMBL3134076 0.61 KCNH2 (0.38) GSK3BTOP2ATOP2BPOLBKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4992546-A Process for preparing 6,8-diazabicyclo[3.2.2]nonane derivatives WARNER-LAMBERT COMPANY (US) 1991-02-12 US disclosed
US-4968799-A Antibacterial agents WARNER-LAMBERT COMPANY (US) 1990-11-06 US disclosed
US-4962108-A A QUIN-4-ONE HAVING THE FOLLOWING RING SUBSTITUENTS; 1-ALKYL OR PHENYL, 3-CARBOXY DERIVATIVE, 6-FLUORO AND 8-BRIDGED N-HETEROCYCLIC RING WARNER-LAMBERT COMPANY (US) 1990-10-09 US disclosed
US-4923879-A CARBOXYLIC ACID DERIVATIVES WITH BRIDGED SIDECHAINS WARNER-LAMBERT COMPANY (US) 1990-05-08 US disclosed
EP-0305744-A2 Quinoline, naphthyridine and benzoxazine-carboxylic acid derivatives and their use as antibacterial agents WARNER-LAMBERT COMPANY (US) 1989-03-08 EP disclosed