SCHEMBL9865852

SCHEMBL9865852

CCNC1CC2CCC(C1)N2c1c(C(=O)O)c(=O)c2cc(F)cc(Cl)c2n1C1CC1

nearest known ligand 0.34

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 2/20 0.34
MAPT P10636 1/20 0.33
KDM4E B2RXH2 2/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
CYP1A2 P05177 1/20 0.32
CCR3 P51677 1/20 0.31
P2RX7 Q99572 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9866155 0.89 KDM4E (0.36) CHRM1MAPTKDM4ESMN1; SMN2CYP1A2
SCHEMBL9865154 0.79 FOXO1 (0.35) CHRM1
Hydrochloric Acid SCHEMBL6005743 0.72 ALDH1A1 (0.48) CHRM1
SCHEMBL3315232 0.70 ALDH1A1 (0.43) CHRM1
SCHEMBL9866818 0.67 GSK3B (0.38)
SCHEMBL9244385 0.67 KCNH2 (0.41) CHRM1MAPTKDM4ESMN1; SMN2CYP1A2
SCHEMBL8324882 0.67 CHRM2 (0.42) KDM4E
SCHEMBL9865560 0.67 TOP2A (0.54) CHRM1MAPTKDM4E
SCHEMBL8866563 0.65
Water SCHEMBL8866780 0.64

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4992546-A Process for preparing 6,8-diazabicyclo[3.2.2]nonane derivatives WARNER-LAMBERT COMPANY (US) 1991-02-12 US disclosed
US-4968799-A Antibacterial agents WARNER-LAMBERT COMPANY (US) 1990-11-06 US disclosed
US-4962108-A A QUIN-4-ONE HAVING THE FOLLOWING RING SUBSTITUENTS; 1-ALKYL OR PHENYL, 3-CARBOXY DERIVATIVE, 6-FLUORO AND 8-BRIDGED N-HETEROCYCLIC RING WARNER-LAMBERT COMPANY (US) 1990-10-09 US disclosed
US-4923879-A CARBOXYLIC ACID DERIVATIVES WITH BRIDGED SIDECHAINS WARNER-LAMBERT COMPANY (US) 1990-05-08 US disclosed
EP-0305744-A2 Quinoline, naphthyridine and benzoxazine-carboxylic acid derivatives and their use as antibacterial agents WARNER-LAMBERT COMPANY (US) 1989-03-08 EP disclosed