SCHEMBL9865624

SCHEMBL9865624

O=C(N=C(NCCCOc1cccc(CN2CCCCC2)c1)Oc1ccccc1)c1ccccc1

nearest known ligand 0.66

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.59
ALDH1A1 P00352 1/20 0.59
HRH2 P25021 1/20 0.58
HRH3 Q9Y5N1 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10675163 0.84 HRH2 (0.67) KDM4EALDH1A1HRH2HRH3
Hydrochloric Acid SCHEMBL10675153 0.83 HRH2 (0.66) KDM4EALDH1A1HRH2HRH3
SCHEMBL10837381 0.83 KDM4E (0.74) KDM4EALDH1A1HRH2HRH3
SCHEMBL9593817 0.83 HRH2 (0.55) KDM4EALDH1A1HRH2HRH3
SCHEMBL9865059 0.81 RAB9A (0.55)
SCHEMBL9593382 0.80 HRH2 (0.52) KDM4EALDH1A1HRH2HRH3
SCHEMBL11086396 0.80 KDM4E (0.75) KDM4EALDH1A1HRH2HRH3
SCHEMBL9865611 0.80 FAAH (0.52) KDM4EALDH1A1HRH2HRH3
SCHEMBL9865618 0.80 FAAH (0.52) KDM4EALDH1A1HRH2HRH3
SCHEMBL11185887 0.79 HRH2 (0.78) KDM4EALDH1A1HRH2HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5021431-A H-1 antagonist, h-2 agonist for treating hypertension, cardiac disease or arterial occlusion HEUMANN PHARMA GMBH & CO. (DE) 1991-06-04 US disclosed