SCHEMBL9866632

SCHEMBL9866632

COC(=O)[C@H](Cc1cccc2ccccc12)NC(=O)[C@H](CC(=O)OC(C)(C)C)NC(=O)c1cccc(NC(=O)c2ccc(C(=N)N)cc2)c1

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 2/20 0.42
ITGA2B P08514 2/20 0.42
CTSS P25774 1/20 0.40
CTSK P43235 1/20 0.40
F10 P00742 11/20 0.40
PLAU P00749 4/20 0.39
F2 P00734 6/20 0.39
PRSS1 P07477 6/20 0.39
PRSS2 P07478 1/20 0.39
PRSS3 P35030 1/20 0.39
PLG P00747 1/20 0.39
PLAT P00750 1/20 0.39
KLKB1 P03952 1/20 0.39
TACR1 P25103 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Iodide SCHEMBL9866617 0.99 ITGB3 (0.41) ITGB3ITGA2BCTSSCTSKF10
SCHEMBL9337488 0.94 ITGB3 (0.47) ITGB3ITGA2BCTSSCTSKPLAU
SCHEMBL9337361 0.90 CTSS (0.44) CTSSCTSKPLAUTACR1
Iodide SCHEMBL9866746 0.90 CTSS (0.44) ITGB3ITGA2BCTSSCTSKF10
Iodide SCHEMBL9866737 0.90 CTSS (0.44) ITGB3ITGA2BCTSSCTSKF10
SCHEMBL9337552 0.88 ITGB3 (0.49) ITGB3ITGA2BF10PLAUF2
Iodide SCHEMBL9337538 0.88 ITGB3 (0.48) ITGB3ITGA2BF10PLAUF2
SCHEMBL9865704 0.85 CTSK (0.44) CTSSCTSKTACR1
SCHEMBL9335862 0.85 CTSS (0.45) CTSSCTSKTACR1
SCHEMBL9339303 0.85 ITGB3 (0.48) ITGB3ITGA2BCTSSCTSKF10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5039805-A Novel benzoic and phenylacetic acid derivatives HOFFMANN-LA ROCHE INC. (US) 1991-08-13 US disclosed