SCHEMBL9865704

SCHEMBL9865704

COC(=O)[C@H](Cc1cccc2ccccc12)NC(=O)[C@H](CC(=O)OC(C)(C)C)NC(=O)c1cccc(NC(=O)OCc2ccccc2)c1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CTSK P43235 2/20 0.44
CTSS P25774 1/20 0.44
CASP3 P42574 1/20 0.44
TACR1 P25103 2/20 0.43
IL1RN P18510 1/20 0.42
ERAP2 Q6P179 1/20 0.42
CTSB P07858 1/20 0.41
CASP1 P29466 1/20 0.41
MGLL Q99685 1/20 0.40
FNTA P49354 1/20 0.40
FNTB P49356 1/20 0.40
ENPP2 Q13822 1/20 0.39
CYP3A4 P08684 1/20 0.39
BACE1 P56817 2/20 0.39
REN P00797 2/20 0.39
MMP8 P22894 1/20 0.39
ALDH1A1 P00352 1/20 0.39
KLK5 Q9Y337 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9865799 0.88 MGLL (0.51) MGLLFNTAFNTBENPP2ALDH1A1
SCHEMBL9866632 0.85 ITGB3 (0.42) CTSKCTSSTACR1
Iodide SCHEMBL9866617 0.85 ITGB3 (0.41) CTSKCTSSTACR1
SCHEMBL9337361 0.84 CTSS (0.44) CTSKCTSSTACR1
SCHEMBL9335862 0.84 CTSS (0.45) CTSKCTSSTACR1FNTACYP3A4
SCHEMBL9867660 0.83 CTSS (0.49) CTSKCTSSCTSB
SCHEMBL9337444 0.83 CTSS (0.44) CTSKCTSSRENKLK5
Iodide SCHEMBL9866746 0.83 CTSS (0.44) CTSKCTSSRENKLK5
SCHEMBL9865501 0.83 CTSS (0.44) CTSKCTSSRENKLK5
SCHEMBL9867667 0.83 CTSS (0.49) CTSKCTSSCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5039805-A Novel benzoic and phenylacetic acid derivatives HOFFMANN-LA ROCHE INC. (US) 1991-08-13 US disclosed