SCHEMBL9866832

SCHEMBL9866832

COc1cc(N)c([N+](=O)[O-])cc1C(=O)NC1CCN(CC2CCCCC2)CC1C

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.54
DRD3 P35462 2/20 0.54
DRD4 P21917 1/20 0.54
HTR4 Q13639 17/20 0.51
KCNH2 Q12809 7/20 0.51
ACHE P22303 2/20 0.51
MLNR O43193 1/20 0.51
ADRB2 P07550 1/20 0.51
CHRM1 P11229 1/20 0.51
ADRA2B P18089 1/20 0.51
ADRA2C P18825 1/20 0.51
CHRM3 P20309 1/20 0.51
SLC6A2 P23975 1/20 0.51
HTR2A P28223 1/20 0.51
SLC6A4 P31645 1/20 0.51
HRH1 P35367 1/20 0.51
OPRK1 P41145 1/20 0.51
HTR2B P41595 1/20 0.51
CHRNA4 P43681 1/20 0.51
HTR3A P46098 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9868098 0.87 MLNR (0.65) DRD2DRD3HTR4KCNH2ACHE
SCHEMBL11180214 0.86 DRD2 (0.72) DRD2DRD3DRD4HTR4KCNH2
SCHEMBL9867444 0.84 DRD4 (0.77) DRD2DRD3DRD4HTR4KCNH2
SCHEMBL9866396 0.81 DRD4 (0.55) DRD2DRD3DRD4HTR4KCNH2
SCHEMBL9865358 0.75 MLNR (0.64) DRD2DRD3HTR4KCNH2ACHE
SCHEMBL9867256 0.75 MLNR (0.84) DRD2DRD3HTR4KCNH2MLNR
SCHEMBL9866959 0.74 DRD4 (0.56) DRD2DRD3DRD4HTR4KCNH2
Hydrochloric Acid SCHEMBL11544323 0.74 HTR4 (0.64) HTR4ACHE
SCHEMBL10722095 0.74 DRD4 (0.73) DRD4HTR4
Denipride SCHEMBL2108137 0.73 DRD2 (0.57) DRD2DRD3DRD4HTR4KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5026858-A Used for treating nausea, vomating, gastrointestinal disorders and centarl nervous system WALTON S.A. (ES) 1991-06-25 US disclosed