SCHEMBL9869324

SCHEMBL9869324

COCOc1c(-c2ccccc2)sc2c(Cc3ccccc3O)nccc12

nearest known ligand 0.31

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HSPA5 P11021 1/20 0.31
CYP1A2 P05177 1/20 0.31
RAB9A P51151 1/20 0.30
CASP3 P42574 1/20 0.30
SENP6 Q9GZR1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9869706 0.84 CYP1A2 (0.34) HSPA5CYP1A2RAB9ACASP3SENP6
SCHEMBL9870823 0.82 HSPA5 (0.38) HSPA5CYP1A2
SCHEMBL9869316 0.74 LMNA (0.40)
SCHEMBL9869471 0.69 BRAF (0.37)
SCHEMBL9869116 0.68 KDM4E (0.43) CYP1A2RAB9A
SCHEMBL9752017 0.61 ALDH1A1 (0.59) HSPA5
SCHEMBL8703013 0.57 MPO (0.49) HSPA5RAB9A
SCHEMBL18969683 0.55 EGFR (0.44) RAB9A
SCHEMBL8745956 0.55 HSPA5 (0.62) HSPA5
SCHEMBL2772333 0.55 TAAR1 (0.54) HSPA5RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5006532-A Enzyme inhibitor; antiinflammatory agents MERCK & CO. INC., INC. (US) 1991-04-09 US disclosed
US-4904672-A Derivatives of 3-hydroxyazabenzo[b]thiophene useful as 5-lipoxygenase inhibitors MERCK & CO., INC. (US) 1990-02-27 US disclosed
US-4767766-A Derivatives of 3-hydroxyazabenzo(B)thiophene useful as 5-lipoxygenase inhibitors MERCK & CO., INC. (US) 1988-08-30 US disclosed