SCHEMBL9869361

SCHEMBL9869361

COc1ccc(CSc2cnccc2C#N)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 2/20 0.56
MAOA P21397 1/20 0.51
PPARG P37231 1/20 0.47
NCOA2 Q15596 1/20 0.47
NCOA1 Q15788 1/20 0.47
NCOA3 Q9Y6Q9 1/20 0.47
ALDH1A1 P00352 3/20 0.46
TDP1 Q9NUW8 2/20 0.46
L3MBTL1 Q9Y468 2/20 0.46
GSK3A P49840 1/20 0.45
GSK3B P49841 1/20 0.45
MEN1 O00255 4/20 0.42
KMT2A Q03164 4/20 0.42
TSHR P16473 3/20 0.42
MAPT P10636 2/20 0.42
KDM4E B2RXH2 1/20 0.42
HPGD P15428 1/20 0.42
HSD17B10 Q99714 1/20 0.42
CYP3A4 P08684 1/20 0.42
APP P05067 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25252466 0.83 MAOB (0.54) MAOBMAOAPPARGNCOA2NCOA1
SCHEMBL30991734 0.83 MAOB (0.54) MAOBMAOAPPARGNCOA2NCOA1
SCHEMBL10470690 0.81 MAOA (0.50) MAOBMAOAPPARGNCOA2NCOA1
SCHEMBL9869356 0.77 SLC22A12 (0.48) MEN1KMT2ATSHRCYP3A4NPC1
SCHEMBL17080256 0.76 MAOB (0.63) MAOBMAOAALDH1A1TDP1L3MBTL1
SCHEMBL29070081 0.76 MAOB (0.63) MAOBMAOAALDH1A1TDP1L3MBTL1
SCHEMBL9869016 0.75 FFAR1 (0.50) GSK3AGSK3BTSHRMAPTKDM4E
SCHEMBL1024806 0.75 KMT2A (0.51) NCOA3ALDH1A1TDP1L3MBTL1MEN1
SCHEMBL9869415 0.74 LMNA (0.53) ALDH1A1L3MBTL1GSK3AGSK3BMEN1
SCHEMBL31294262 0.74 MAOB (0.67) MAOBMAOAPPARGNCOA2NCOA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5006532-A Enzyme inhibitor; antiinflammatory agents MERCK & CO. INC., INC. (US) 1991-04-09 US disclosed
US-4904672-A Derivatives of 3-hydroxyazabenzo[b]thiophene useful as 5-lipoxygenase inhibitors MERCK & CO., INC. (US) 1990-02-27 US disclosed
US-4767766-A Derivatives of 3-hydroxyazabenzo(B)thiophene useful as 5-lipoxygenase inhibitors MERCK & CO., INC. (US) 1988-08-30 US disclosed