SCHEMBL9870867

SCHEMBL9870867

Cc1cc(-c2ccccc2F)n2ccnc2n1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 3/20 0.42
GABRG2 P18507 3/20 0.42
GABRB3 P28472 3/20 0.42
GABRA3 P34903 3/20 0.42
PDE2A O00408 2/20 0.41
CCNE2 O96020 2/20 0.40
CCNE1 P24864 2/20 0.40
CDK2 P24941 2/20 0.40
MAP2K1 Q02750 1/20 0.39
GABRA5 P31644 2/20 0.39
GABRA2 P47869 1/20 0.39
FLT1 P17948 1/20 0.38
CDK8 P49336 1/20 0.38
CDK9 P50750 1/20 0.38
LIMK1 P53667 1/20 0.38
ROCK1 Q13464 1/20 0.38
CLK4 Q9HAZ1 1/20 0.38
ADORA2A P29274 2/20 0.38
MAPT P10636 2/20 0.38
KDM4E B2RXH2 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9870091 0.79 KDM4E (0.55) GABRA1GABRG2GABRB3GABRA3MAP2K1
SCHEMBL9869845 0.79 EGLN2 (0.50) GABRA1GABRG2GABRB3GABRA3CCNE2
SCHEMBL11009148 0.73 BACE1 (0.49) GABRA1GABRG2GABRB3GABRA3PDE2A
SCHEMBL11009952 0.72 CYP2A6 (0.46) GABRA1GABRG2GABRB3GABRA3GABRA5
SCHEMBL7224559 0.71 GABRA1 (0.70) GABRA1GABRG2GABRB3GABRA3GABRA5
SCHEMBL9870239 0.70 KDM4E (0.43) PDE2ACDK2CDK9MAPTKDM4E
SCHEMBL259043 0.69 KDM4E (0.50) PDE2AMAPTKDM4E
SCHEMBL3704252 0.69 ADORA2A (0.41) GABRA1GABRG2GABRB3GABRA3CCNE2
SCHEMBL9869878 0.69 KDM4E (0.44) PDE2AMAPTKDM4EMAPK1
SCHEMBL3707772 0.69 KDM4E (0.43) GABRA1GABRG2GABRB3GABRA3CCNE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5037980-A Anxiolytic agents, hypotensive agents AMERICAN CYANAMID COMPANY (US) 1991-08-06 US disclosed