SCHEMBL9873422

SCHEMBL9873422

COC(=O)c1c(F)c(F)c(C2(C(=O)OC(c3ccccc3)c3ccccc3)CC2)c(F)c1F

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.38
TP53 P04637 1/20 0.38
ESR1 P03372 1/20 0.37
ESR2 Q92731 1/20 0.37
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA7 P43166 1/20 0.36
CA9 Q16790 1/20 0.36
CA14 Q9ULX7 1/20 0.36
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 2/20 0.36
LMNA P02545 1/20 0.36
HPGD P15428 1/20 0.36
TSHR P16473 2/20 0.34
CYP3A4 P08684 2/20 0.33
CYP2D6 P10635 2/20 0.33
CYP2C9 P11712 2/20 0.33
MAPK1 P28482 1/20 0.33
GAA P10253 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9872913 0.76 KMT2A (0.41) KMT2ATP53ESR1ESR2CA12
SCHEMBL9873993 0.76 TSHR (0.42) CA12CA1CA2CA7CA9
SCHEMBL9872562 0.75 MAPK1 (0.39) KMT2ATP53ESR1ESR2KDM4E
SCHEMBL9873671 0.74 CRHBP (0.45) KMT2ATP53ESR1ESR2CA12
SCHEMBL9874015 0.74 LMNA (0.40) KMT2ATP53KDM4EALDH1A1LMNA
SCHEMBL18527167 0.68 ESR1 (0.47) KMT2AESR1ESR2KDM4EALDH1A1
SCHEMBL11000173 0.67 KMT2A (0.57) KMT2AESR1ESR2KDM4EALDH1A1
SCHEMBL13545931 0.66 ESR1 (0.72) KMT2AESR1ESR2CA12CA1
SCHEMBL505248 0.66 LMNA (0.57) KMT2ATP53CA12CA1CA2
SCHEMBL28947855 0.66 ESR1 (0.45) KMT2AESR1ESR2KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4990508-A Reduced side effects TOYAMA CHEMICAL CO., LTD. (JP) 1991-02-05 US disclosed