SCHEMBL9879130

SCHEMBL9879130

COCc1nc(N)[nH]c(=O)c1C

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TYMS P04818 1/20 0.43
XDH P47989 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
NPSR1 Q6W5P4 1/20 0.39
MAPK1 P28482 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
HTT P42858 1/20 0.39
PNP P00491 1/20 0.37
CYP1A2 P05177 1/20 0.36
KMT2A Q03164 1/20 0.35
HIF1A Q16665 1/20 0.35
TYMP P19971 1/20 0.34
MAPT P10636 1/20 0.34
CDK1 P06493 1/20 0.34
CDK4 P11802 1/20 0.34
CDK2 P24941 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9878825 0.76 HTT (0.70) XDHL3MBTL1SMN1; SMN2HTTKMT2A
SCHEMBL9879126 0.71 L3MBTL1 (0.46) TYMSXDHL3MBTL1NPSR1MAPK1
SCHEMBL718210 0.70 NPSR1 (0.52) XDHL3MBTL1NPSR1MAPK1PNP
SCHEMBL12956972 0.70 CDK1 (0.52) TYMSXDHL3MBTL1NPSR1PNP
SCHEMBL2343355 0.68 PNP (0.59) PNPKMT2AMAPT
SCHEMBL18294954 0.67 SMN1; SMN2 (0.55) L3MBTL1MAPK1SMN1; SMN2HTTCYP1A2
SCHEMBL9879338 0.67 HSP90AA1 (0.38) L3MBTL1NPSR1SMN1; SMN2CYP1A2KMT2A
SCHEMBL9878974 0.67 MEN1 (0.51) MAPK1KMT2AMAPT
SCHEMBL10618579 0.65 NOS1 (0.68) KMT2AMAPT
SCHEMBL22354697 0.64 ALDH1A1 (0.43) TYMSXDHNPSR1MAPK1PNP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991018887-A1 DIAMINOPYRIMIDINE COMPOUNDS SMITHKLINE BEECHAM INTERCREDIT B.V. (NL) 1991-12-12 WO disclosed