SCHEMBL9880967

SCHEMBL9880967

CCC(CC(C)C)c1ccsc1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.38
IDO1 P14902 1/20 0.33
TDO2 P48775 1/20 0.33
CHRNB2 P17787 1/20 0.32
CHRNB4 P30926 1/20 0.32
CHRNA3 P32297 1/20 0.32
CHRNA4 P43681 1/20 0.32
TAS1R3 Q7RTX0 1/20 0.31
TAS1R1 Q7RTX1 1/20 0.31
CYP17A1 P05093 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
SLC6A2 P23975 1/20 0.31
SLC6A4 P31645 1/20 0.31
SLC6A3 Q01959 1/20 0.31
KCNH2 Q12809 1/20 0.31
DRD2 P14416 1/20 0.30
DRD3 P35462 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12464829 0.86 ALOX5 (0.39) ALOX5IDO1TDO2CHRNB2CHRNB4
SCHEMBL9883273 0.80 SLC6A2 (0.43) ALOX5TAS1R3TAS1R1CYP3A4CYP2D6
SCHEMBL22995905 0.78 ALOX5 (0.39) ALOX5IDO1TDO2CHRNB2CHRNB4
SCHEMBL2992960 0.78 ALOX5 (0.39) ALOX5IDO1TDO2CHRNB2CHRNB4
SCHEMBL13848615 0.78 CHRNB2 (0.36) ALOX5IDO1TDO2CHRNB2CHRNB4
SCHEMBL14516277 0.76 NR1I2 (0.41) ALOX5IDO1TDO2CHRNB2CHRNB4
SCHEMBL7874405 0.75
SCHEMBL20987465 0.75 ALOX5 (0.34) ALOX5CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL27818681 0.74 ALOX5 (0.39) ALOX5IDO1TDO2CHRNB2CHRNB4
SCHEMBL12462086 0.74 ALOX5 (0.36) ALOX5IDO1TDO2CHRNB2CHRNB4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20170196862-A2 MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR VERTEX PHARMACEUTICALS INCORPORATED (US) 2017-07-13 US disclosed
US-20120135984-A1 DUAL-ACTION INHBITORS AND METHODS OF USING SAME AERIE PHARMACEUTICALS, INC. 2012-05-31 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120135984-A1 DUAL-ACTION INHBITORS AND METHODS OF USING SAME SLC6A2, ROCK2, SLC6A4 ALOX5 2859/4885IDO1 104/4885TDO2 819/4885
US-20170196862-A2 MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR CFTR, SCNN1B, SLC26A4 ALOX5 3465/4885IDO1 4683/4885TDO2 4435/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.