SCHEMBL989934

SCHEMBL989934

C=C(CBr)c1ccc(OC)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 1/20 0.60
MAPT P10636 2/20 0.50
NR1I2 O75469 1/20 0.50
MAOA P21397 1/20 0.49
MAOB P27338 1/20 0.49
CES2 O00748 1/20 0.48
CES1 P23141 1/20 0.48
CA1 P00915 5/20 0.47
CA2 P00918 5/20 0.47
CA12 O43570 1/20 0.46
CA7 P43166 1/20 0.46
CA9 Q16790 1/20 0.46
CA14 Q9ULX7 1/20 0.46
MEN1 O00255 1/20 0.46
LMNA P02545 1/20 0.46
MAPK1 P28482 1/20 0.46
RAB9A P51151 1/20 0.46
KMT2A Q03164 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
RXFP1 Q9HBX9 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14407542 0.81 NR1I2 (0.52) GSK3BMAPTNR1I2MAOAMAOB
SCHEMBL5085228 0.81 NR1I2 (0.63) GSK3BMAPTNR1I2MAOAMAOB
SCHEMBL20716157 0.80 NQO1 (0.54) MAOBLMNARAB9AKMT2ANPSR1
SCHEMBL13962133 0.79 CA1 (0.50) MAPTNR1I2MAOAMAOBCA1
SCHEMBL8552180 0.79 LMNA (0.51) GSK3BMAPTNR1I2MAOAMAOB
SCHEMBL16795750 0.79 MAPT (0.50) GSK3BMAPTNR1I2MAOAMAOB
SCHEMBL24148257 0.77 MAPT (0.62) GSK3BMAPTCES2CES1CA1
SCHEMBL16795587 0.77 LMNA (0.55) GSK3BMAPTMEN1LMNARAB9A
SCHEMBL9364978 0.77 CES2 (0.55) MAOAMAOBCES2CES1MEN1
SCHEMBL202055 0.75 GSK3B (1.00) GSK3BMAPTCES2CES1CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2585457-B1 Alkaloid aminoester derivatives and medicinal composition thereof CHIESI FARMA SPA (IT) 2015-07-22 EP disclosed
EP-2862856-A1 AROMATIC HETEROCYCLIC COMPOUND Mitsubishi Tanabe Pharma Corporation (JP) 2015-04-22 EP disclosed
EP-2480080-A1 PYRIDO[3,4-B]INDOLES AND METHODS OF USE Medivation Technologies, Inc. (US) 2012-08-01 EP disclosed
EP-2338334-A1 Pesticides and uses thereof Dow AgroSciences LLC (US) 2011-06-29 EP disclosed
WO-2011038163-A1 PYRIDO[3,4-B]INDOLES AND METHODS OF USE MEDIVATION TECHNOLOGIES, INC. (US) 2011-03-31 WO disclosed
EP-2274307-A1 BRIDGED HETEROCYCLIC COMPOUNDS AND METHODS OF USE Medivation Technologies, Inc. (US) 2011-01-19 EP disclosed
WO-2009120720-A1 BRIDGED HETEROCYCLIC COMPOUNDS AND METHODS OF USE MEDIVATION TECHNOLOGIES,INC. (US) 2009-10-01 WO disclosed