SCHEMBL8552180

SCHEMBL8552180

C=C(COC)c1ccc(OC)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.51
NR1I2 O75469 1/20 0.50
MAPT P10636 1/20 0.50
MAOA P21397 1/20 0.49
MAOB P27338 1/20 0.49
CES2 O00748 1/20 0.48
CES1 P23141 1/20 0.48
CA1 P00915 5/20 0.47
CA2 P00918 5/20 0.47
CA12 O43570 1/20 0.46
CA7 P43166 1/20 0.46
CA9 Q16790 1/20 0.46
CA14 Q9ULX7 1/20 0.46
GSK3B P49841 1/20 0.46
HDAC3 O15379 1/20 0.46
HDAC4 P56524 1/20 0.46
HDAC1 Q13547 1/20 0.46
HDAC7 Q8WUI4 1/20 0.46
HDAC2 Q92769 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5085228 0.81 NR1I2 (0.63) LMNANR1I2MAPTMAOAMAOB
SCHEMBL14407542 0.81 NR1I2 (0.52) LMNANR1I2MAPTMAOAMAOB
SCHEMBL22561008 0.81 KDM4E (0.49) LMNAL3MBTL1MAPTALDH1A1SMN1; SMN2
SCHEMBL16795750 0.79 MAPT (0.50) LMNANR1I2MAPTMAOAMAOB
SCHEMBL13962133 0.79 CA1 (0.50) NR1I2MAPTMAOAMAOBCA1
SCHEMBL8554384 0.79 MAOA (0.50) LMNAL3MBTL1MAPTMAOAMAOB
SCHEMBL989934 0.79 GSK3B (0.60) LMNANR1I2MAPTMAOAMAOB
SCHEMBL10855469 0.79 CYP3A4 (0.41) LMNAMAPTMAOAALDH1A1PRSS1
SCHEMBL8557285 0.77 CES2 (0.55) LMNAMAOAMAOBCES2CES1
SCHEMBL20446944 0.77 CA1 (0.65) L3MBTL1MAPTCA1CA2SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0861245-A1 PIPERIDINE AND TETRAHYDROPYRIDINE DERIVATIVES MERCK SHARP & DOHME LTD. (GB) 1998-09-02 EP disclosed
WO-1997019073-A1 PIPERIDINE AND TETRAHYDROPYRIDINE DERIVATIVES MERCK SHARP & DOHME LIMITED (GB) 1997-05-29 WO disclosed