SCHEMBL9901522

SCHEMBL9901522

CCOC(=O)C=C(ON(NC(=O)OCc1ccccc1)C(=N)C1CCC(COS(=O)(=O)c2ccc(C)cc2)(COS(=O)(=O)c2ccc(C)cc2)CC1)C(=O)OCC

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CA1 P00915 5/20 0.35
CA2 P00918 5/20 0.35
TGM2 P21980 4/20 0.35
F13A1 P00488 3/20 0.35
TGM1 P22735 3/20 0.35
P2RX7 Q99572 5/20 0.34
HPN P05981 1/20 0.32
ST14 Q9Y5Y6 1/20 0.32
LMNA P02545 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
POLB P06746 1/20 0.32
ELANE P08246 1/20 0.32
MMP2 P08253 1/20 0.32
MMP9 P14780 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9900927 0.82 KDM1A (0.37) LMNA
SCHEMBL9942922 0.78 F13A1 (0.37) CA1CA2TGM2F13A1TGM1
SCHEMBL9900865 0.68 LMNA (0.43) CA1CA2P2RX7HPNST14
SCHEMBL28328057 0.66 LMNA (0.48) CA1CA2P2RX7LMNAELANE
SCHEMBL9942900 0.66 CTSL (0.44) CA1CA2P2RX7LMNA
SCHEMBL23540158 0.66 APP (0.50) CA1CA2TGM2F13A1TGM1
SCHEMBL5528333 0.65 TLR2 (0.41)
SCHEMBL13924823 0.64 NR1H4 (0.49) TGM2F13A1TGM1LMNAMEN1
SCHEMBL51559 0.63 CTSS (0.38)
SCHEMBL144613 0.63 P2RX7 (0.41) CA1CA2TGM2F13A1TGM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2649077-A1 HIV INTEGRASE INHIBITORS Bristol-Myers Squibb Company (US) 2013-10-16 EP disclosed
WO-2012078834-A1 HIV INTEGRASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2012-06-14 WO disclosed