SCHEMBL990795

SCHEMBL990795

C=C(C)CC(O)(CCN(C(=O)O)C(C)(C)C#Cc1ccc(F)cc1)c1ccccc1

nearest known ligand 0.37

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 2/20 0.37
NR1H2 P55055 3/20 0.35
HTT P42858 1/20 0.32
MAPT P10636 1/20 0.32
KCNN4 O15554 2/20 0.32
ALOX5 P09917 1/20 0.31
FFAR1 O14842 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL992158 0.90 HSD11B1 (0.35) HSD11B1NR1H2HTTMAPTKCNN4
SCHEMBL991395 0.80 CYP2C19 (0.34) HTTMAPT
SCHEMBL12950521 0.75 KCNN4 (0.36) NR1H2MAPTKCNN4
SCHEMBL116411 0.75 OPRM1 (0.34) MAPT
SCHEMBL991891 0.70 ALDH1A1 (0.35) NR1H2HTTMAPTKCNN4
SCHEMBL11922654 0.68 SMN1; SMN2 (0.57)
SCHEMBL991959 0.66 OGT (0.40) HSD11B1
SCHEMBL11055846 0.66 CYP2C19 (0.48) HTTKCNN4
SCHEMBL1431288 0.65 ALOX5 (0.36) ALOX5
SCHEMBL1431286 0.65 ALOX5 (0.36) ALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2440537-A1 CYCLIC INHIBITORS OF 11BETA-HYDROXYSTEROID DEHYDROGENASE 1 BASED ON THE 1,3 -OXAZINAN- 2 -ONE STRUCTURE Vitae Pharmaceuticals, Inc. (US) 2012-04-18 EP disclosed
WO-2011011123-A1 CYCLIC INHIBITORS OF 11BETA-HYDROXYSTEROID DEHYDROGENASE 1 BASED ON THE 1,3 -OXAZINAN- 2 -ONE STRUCTURE VITAE PHARMACEUTICALS, INC. (US) 2011-01-27 WO disclosed