SCHEMBL99089

SCHEMBL99089

CC(=O)Nc1ccc(Br)cc1-c1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.56
NPSR1 Q6W5P4 2/20 0.51
POLB P06746 2/20 0.51
LMNA P02545 2/20 0.51
KDM4E B2RXH2 3/20 0.50
HDAC1 Q13547 2/20 0.50
APOBEC3A P31941 1/20 0.50
GFER P55789 1/20 0.50
APOBEC3G Q9HC16 1/20 0.50
HDAC3 O15379 1/20 0.49
HDAC2 Q92769 1/20 0.49
RXFP1 Q9HBX9 2/20 0.49
HTT P42858 2/20 0.47
PTGDR2 Q9Y5Y4 1/20 0.47
PTGFR P43088 1/20 0.46
HIF1A Q16665 1/20 0.45
NPC1 O15118 2/20 0.45
RAB9A P51151 2/20 0.45
MAPT P10636 2/20 0.45
AKR1C3 P42330 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30307389 1.00 ALDH1A1 (0.56) ALDH1A1NPSR1POLBLMNAKDM4E
SCHEMBL15823673 0.87 ALDH1A1 (0.57) ALDH1A1NPSR1POLBLMNARXFP1
SCHEMBL28724549 0.86 ALDH1A1 (0.62) ALDH1A1POLBLMNAKDM4EHDAC1
SCHEMBL29572629 0.86 ALDH1A1 (0.62) ALDH1A1POLBLMNAKDM4EHDAC1
SCHEMBL17206261 0.85 KDM4E (0.55) ALDH1A1POLBLMNAKDM4EHDAC1
SCHEMBL3907636 0.84 ALDH1A1 (0.51) ALDH1A1NPSR1POLBLMNARXFP1
SCHEMBL20194476 0.83 HDAC1 (0.66) ALDH1A1NPSR1POLBLMNAKDM4E
SCHEMBL11187279 0.82 HDAC7 (0.54) ALDH1A1POLBLMNAKDM4EHDAC1
SCHEMBL17209129 0.81 MAPT (0.54) ALDH1A1POLBKDM4EHDAC1APOBEC3A
SCHEMBL21244213 0.81 KDM4E (0.64) NPSR1LMNAKDM4EHDAC1APOBEC3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9072734-B2 Quaternary ammonium salt compounds TEIJIN PHARMA LIMITED (JP) 2015-07-07 US disclosed
EP-2426121-A1 QUATERNARY AMMONIUM SALT COMPOUND Teijin Pharma Limited (JP) 2012-03-07 EP disclosed
US-20120046467-A1 QUATERNARY AMMONIUM SALT COMPOUNDS TEIJIN PHARMA LIMITED (JP) 2012-02-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120046467-A1 QUATERNARY AMMONIUM SALT COMPOUNDS ADRB2, AGTR2, ADRB3 ALDH1A1 1896/4885NPSR1 253/4885POLB 3291/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.