SCHEMBL9911403

SCHEMBL9911403

Cc1nncn1-c1ccc(C2CC2)cc1Cl

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GABRG2 P18507 2/20 0.39
GABRB3 P28472 2/20 0.39
GABRA5 P31644 2/20 0.39
SMURF1 Q9HCE7 4/20 0.36
SMURF2 Q9HAU4 1/20 0.36
SLC6A2 P23975 6/20 0.34
SLC6A4 P31645 6/20 0.34
SLC6A3 Q01959 6/20 0.34
CYP2D6 P10635 5/20 0.34
KCNH2 Q12809 4/20 0.34
PDE2A O00408 1/20 0.34
CYP11B2 P19099 1/20 0.32
OPRM1 P35372 1/20 0.31
FASN P49327 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9911410 0.84 GABRG2 (0.37) GABRG2GABRB3GABRA5SMURF1SMURF2
SCHEMBL17069753 0.69 SLC22A12 (0.41) SLC6A4CYP2D6
SCHEMBL12693003 0.69 ESR2 (0.39) SLC6A2SLC6A4SLC6A3
SCHEMBL879247 0.67 SLC6A2 (0.57) SMURF1SMURF2SLC6A2SLC6A4SLC6A3
SCHEMBL17260097 0.66 SMURF1 (0.59) SMURF1SMURF2
SCHEMBL9610090 0.66 L3MBTL1 (0.40) GABRG2GABRB3GABRA5SMURF1KCNH2
SCHEMBL879149 0.65 SMURF1 (0.34) GABRG2GABRB3GABRA5SMURF1SMURF2
SCHEMBL9870878 0.64 SLC6A2 (0.58) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2
SCHEMBL9912504 0.63 SLC6A2 (0.57) SMURF1SMURF2SLC6A2SLC6A4SLC6A3
SCHEMBL3107895 0.63 GABRG2 (0.34) GABRG2GABRB3GABRA5KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8198458-B2 Non-nucleoside reverse transcriptase inhibitors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-06-12 US disclosed
US-20090143370-A1 Non-nucleoside Reverse Transcriptase Inhibitors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-06-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090143370-A1 Non-nucleoside Reverse Transcriptase Inhibitors RTF1, POLR1A, POLR1E GABRG2 4463/4885GABRB3 4569/4885GABRA5 4630/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.