SCHEMBL9912203

SCHEMBL9912203

Cc1noc(-c2cccc(-c3cc(NCCc4ccc(O)cc4)nc(O)n3)c2)n1

nearest known ligand 0.66

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PTGDR Q13258 15/20 0.66
PIK3CA P42336 2/20 0.42
PIK3CB P42338 2/20 0.42
PIK3CG P48736 2/20 0.42
ALDH1A1 P00352 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
TP53 P04637 1/20 0.37
MAPT P10636 1/20 0.37
HRH1 P35367 1/20 0.37
HRH4 Q9H3N8 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4511595 0.80 PTGDR (1.00) PTGDR
SCHEMBL13894999 0.78 ALDH1A1 (0.47) PTGDRPIK3CAPIK3CBPIK3CGALDH1A1
SCHEMBL9912189 0.77 BCHE (0.47) PTGDRPIK3CAPIK3CBPIK3CGALDH1A1
SCHEMBL9912204 0.77 PTGDR (0.56) PTGDRPIK3CAPIK3CBPIK3CGALDH1A1
SCHEMBL9912237 0.76 PTGDR (0.52) PTGDRPIK3CAPIK3CBPIK3CGALDH1A1
SCHEMBL9912281 0.76 BRAF (0.61) PTGDRALDH1A1SMN1; SMN2TP53MAPT
SCHEMBL9912276 0.75 PTGDR (0.63) PTGDRPIK3CAPIK3CBPIK3CGALDH1A1
SCHEMBL13895056 0.75 ALDH1A1 (0.44) PTGDRALDH1A1SMN1; SMN2
SCHEMBL9912208 0.73 PTGDR (0.57) PTGDRPIK3CAPIK3CBPIK3CGALDH1A1
SCHEMBL9912205 0.73 PTGDR (0.52) PTGDRPIK3CAPIK3CBPIK3CGALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8193183-B2 2,6-substituted-4-monosubstitutedamino-pyrimidine as prostaglandin D2 receptor antagonists AVENTIS PHARMACEUTICALS INC. (US) 2012-06-05 US disclosed