SCHEMBL9912276

SCHEMBL9912276

N#CCc1cccc(-c2cc(NCCc3ccc(O)cc3)nc(O)n2)c1

nearest known ligand 0.63

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PTGDR Q13258 13/20 0.63
MMP3 P08254 1/20 0.51
ALDH1A1 P00352 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
PIK3CA P42336 2/20 0.42
PIK3CB P42338 2/20 0.42
PIK3CG P48736 2/20 0.42
ADORA2A P29274 1/20 0.42
HRH1 P35367 1/20 0.39
HRH4 Q9H3N8 1/20 0.39
USP7 Q93009 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13894999 0.85 ALDH1A1 (0.47) PTGDRALDH1A1SMN1; SMN2PIK3CAPIK3CB
SCHEMBL9912189 0.84 BCHE (0.47) PTGDRALDH1A1SMN1; SMN2PIK3CAPIK3CB
SCHEMBL9912207 0.81 PTGDR (0.51) PTGDRMMP3PIK3CAPIK3CBPIK3CG
SCHEMBL9912210 0.80 ALDH1A1 (0.44) PTGDRALDH1A1SMN1; SMN2PIK3CAPIK3CB
SCHEMBL9912204 0.80 PTGDR (0.56) PTGDRALDH1A1SMN1; SMN2PIK3CAPIK3CB
SCHEMBL9912237 0.79 PTGDR (0.52) PTGDRALDH1A1SMN1; SMN2PIK3CAPIK3CB
SCHEMBL4491413 0.77 PTGDR (1.00) PTGDR
SCHEMBL9912281 0.77 BRAF (0.61) PTGDRALDH1A1SMN1; SMN2
SCHEMBL9912208 0.77 PTGDR (0.57) PTGDRALDH1A1SMN1; SMN2PIK3CAPIK3CB
SCHEMBL9912203 0.75 PTGDR (0.66) PTGDRALDH1A1SMN1; SMN2PIK3CAPIK3CB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8193183-B2 2,6-substituted-4-monosubstitutedamino-pyrimidine as prostaglandin D2 receptor antagonists AVENTIS PHARMACEUTICALS INC. (US) 2012-06-05 US disclosed