SCHEMBL9912437

SCHEMBL9912437

O=C(CO)Nc1ccc(C(=O)O)cc1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 2/20 0.56
CA2 P00918 2/20 0.56
CA9 Q16790 2/20 0.56
ALDH1A1 P00352 3/20 0.53
CSNK2A2 P19784 1/20 0.53
CSNK2A1 P68400 1/20 0.53
CYP1A2 P05177 1/20 0.53
CYP2C9 P11712 1/20 0.53
MEN1 O00255 2/20 0.52
KMT2A Q03164 2/20 0.52
MITF O75030 1/20 0.52
CA1 P00915 1/20 0.51
GAA P10253 1/20 0.50
POLB P06746 1/20 0.50
FFAR1 O14842 1/20 0.50
TP53 P04637 1/20 0.50
TSHR P16473 1/20 0.50
HSD17B10 Q99714 1/20 0.49
STAT3 P40763 1/20 0.49
HPGD P15428 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2352584 0.87 MEN1 (0.56) ALDH1A1MEN1KMT2AMITFGAA
SCHEMBL2843886 0.83 CA12 (0.56) CA12CA2CA9ALDH1A1CYP1A2
SCHEMBL3911049 0.82 CA12 (0.54) CA12CA2CA9ALDH1A1CYP1A2
SCHEMBL2344100 0.82 CA12 (0.54) CA12CA2CA9ALDH1A1CYP1A2
SCHEMBL925339 0.82 MAPT (0.64) ALDH1A1MEN1KMT2AGAAPOLB
SCHEMBL216113 0.82 CA12 (0.54) CA12CA2CA9ALDH1A1CYP1A2
SCHEMBL2940113 0.82 ALDH1A1 (0.65) CA12CA2CA9ALDH1A1CYP1A2
SCHEMBL6691641 0.82 MITF (0.55) CA12CA2CA9ALDH1A1CYP1A2
SCHEMBL1663647 0.82 CA2 (0.58) CA12CA2CA9ALDH1A1CYP1A2
SCHEMBL1395934 0.82 ALDH1A1 (0.71) CA12CA2CA9ALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116478131-A 2, 5-disubstituted and 2,5, 6-trisubstituted 3-methylpyrazines as allosteric SHP2 inhibitors 锐新医药公司 2023-07-25 CN disclosed
CN-116478132-A 2, 5-disubstituted and 2,5, 6-trisubstituted 3-methylpyrazines as allosteric SHP2 inhibitors 锐新医药公司 2023-07-25 CN disclosed
CN-110914416-B Microorganism and method for producing cannabinoids and cannabinoid derivatives 加州大学董事会 2023-07-21 CN disclosed
CN-115397809-A Macrocyclic pantetheine derivatives and uses thereof 彗星医疗股份有限公司 2022-11-25 CN disclosed
CN-108135871-B Amine naphthoquinone compounds and pharmaceutical compositions for blocking ubiquitination-proteasome system in diseases 博蔚医药生物科技股份有限公司 2022-11-04 CN disclosed
CN-114641466-A Sulfonylurea derivatives and use thereof 诺瑟拉有限公司 2022-06-17 CN disclosed
CN-108366979-B Compounds and pharmaceutical compositions relating to ubiquitination-proteasome system 博蔚医药生物科技股份有限公司 2021-10-01 CN disclosed
CN-108473497-B EP4 antagonists 卫材R&D 管理有限公司 2021-09-10 CN disclosed
CN-111201232-A ATF3 inducing compounds 台北医学大学 2020-05-26 CN disclosed
CN-110840870-A Use of selective androgen receptor modulators for the treatment of metastatic and refractory breast cancer GTX公司 2020-02-28 CN disclosed
CN-102153481-B Application of thionyl chloride and alcohol as selective deacylation reagents for N-aryl fatty amide or N-heterocyclic fatty amide UNIV SOUTHWEST 2013-09-18 CN disclosed
US-8198458-B2 Non-nucleoside reverse transcriptase inhibitors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-06-12 US disclosed
CN-102153481-A Application of thionyl chloride and alcohol as selective deacylation reagents for N-aryl fatty amide or N-heterocyclic fatty amide UNIV SOUTHWEST 2011-08-17 CN disclosed
US-7517998-B2 Benzothiazole or benzothiazine derivative of dipyrido(2,3;b:2',3'-e) diazepin-6-one; viricide against human t-cell leukemia/lymphoma virus BOEHRINGER INGELHEIM INTERNATIONAL GMBH 2009-04-14 US disclosed