SCHEMBL9924065

SCHEMBL9924065

CCOC(=O)N[C@H]1CC[C@H](N/C(=N\C(=O)c2ccc(F)c(F)c2)NCc2ccc(F)cc2Cl)CC1

nearest known ligand 0.42

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 19/20 0.42
CYP2D6 P10635 1/20 0.41
PKM P14618 1/20 0.41
CYP2C19 P33261 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9923858 0.92 ALDH1A1 (0.41) P2RX7
SCHEMBL9923859 0.91 CHRM1 (0.41)
SCHEMBL9924270 0.91 HPGD (0.40) P2RX7
SCHEMBL9924251 0.90 CYP2D6 (0.41) P2RX7CYP2D6PKMCYP2C19
SCHEMBL9924064 0.90 CHRM1 (0.40) P2RX7
SCHEMBL9924271 0.88 P2RX7 (0.43) P2RX7
SCHEMBL9924063 0.86 SMN1; SMN2 (0.43)
SCHEMBL9924273 0.86 CHRM1 (0.41)
SCHEMBL9924274 0.86 CHRM1 (0.41)
SCHEMBL9924067 0.85 SMN1; SMN2 (0.43) P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9169199-B2 Cycloalkyl guanidine F1F0-ATPase inhibitors and therapeutic uses thereof LYCERA CORPORATION (US) 2015-10-27 US disclosed
WO-2012078867-A2 CYCLOALKYL GUANIDINE F1F0-ATPASE INHIBITORS AND THERAPEUTIC USES THEREOF LYCERA CORPORATION (US) 2012-06-14 WO disclosed