SCHEMBL9952593

SCHEMBL9952593

Nc1nc2ccc(-c3cncc(N4CCOC4=O)c3)cc2c(=O)n1-c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PI4KA P42356 14/20 0.47
PIK3CG P48736 11/20 0.47
TNKS O95271 1/20 0.43
CYP11B2 P19099 1/20 0.42
CCNC P24863 1/20 0.39
CDK8 P49336 1/20 0.39
HCAR1 Q9BXC0 1/20 0.36
HTR1A P08908 1/20 0.35
DRD2 P14416 1/20 0.35
HTR1D P28221 1/20 0.35
HTR1B P28222 1/20 0.35
HTR2A P28223 1/20 0.35
HTR7 P34969 1/20 0.35
DRD3 P35462 1/20 0.35
HTR2B P41595 1/20 0.35
HTR6 P50406 1/20 0.35
KCNH2 Q12809 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Formic Acid SCHEMBL9954795 0.95 PI4KA (0.44) PI4KAPIK3CGTNKSCYP11B2CCNC
SCHEMBL10288787 0.82 PI4KA (0.50) PI4KAPIK3CGCYP11B2HCAR1
SCHEMBL9954049 0.79 PI4KA (0.53) PI4KAPIK3CGHCAR1
Formic Acid SCHEMBL9954566 0.78 PI4KA (0.47) PI4KAPIK3CGCYP11B2HCAR1
SCHEMBL9954693 0.77 PIM1 (0.46) PI4KAPIK3CGCYP11B2
SCHEMBL10288780 0.76 PI4KA (0.52) PI4KAPIK3CGHCAR1
SCHEMBL9953679 0.76 PI4KA (0.51) PI4KAPIK3CGCYP11B2HCAR1
SCHEMBL9954428 0.76 PI4KA (0.56) PI4KAPIK3CG
SCHEMBL9955619 0.76 PI4KA (0.56) PI4KAPIK3CGCYP11B2
SCHEMBL9953943 0.76 PI4KA (0.59) PI4KAPIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012087938-A1 QUINAZOLINONE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-06-28 WO disclosed
WO-2012087938-A1 QUINAZOLINONE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-06-28 WO disclosed